Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 6429
TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 50397656BDBM50397656(CHEMBL2181745 | US8796280, 17)
Affinity DataKi:  380nM ΔG°:  -36.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128328BDBM128328(US8796280, 18)
Affinity DataKi:  400nM ΔG°:  -36.5kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128314BDBM128314(US8796280, 3)
Affinity DataKi:  450nM ΔG°:  -36.2kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128329BDBM128329(US8796280, 19)
Affinity DataKi:  470nM ΔG°:  -36.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128330BDBM128330(US8796280, 20)
Affinity DataKi:  480nM ΔG°:  -36.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128331BDBM128331(US8796280, 21)
Affinity DataKi:  590nM ΔG°:  -35.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128332BDBM128332(US8796280, 22)
Affinity DataKi:  620nM ΔG°:  -35.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128333BDBM128333(US8796280, 23)
Affinity DataKi:  700nM ΔG°:  -35.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128334BDBM128334(US8796280, 24)
Affinity DataKi:  720nM ΔG°:  -35.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128335BDBM128335(US8796280, 25)
Affinity DataKi:  850nM ΔG°:  -34.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128336BDBM128336(US8796280, 26)
Affinity DataKi:  950nM ΔG°:  -34.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128312BDBM128312(US8796280, 1)
Affinity DataKi:  1.01E+3nM ΔG°:  -34.2kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128313BDBM128313(US8796280, 2)
Affinity DataKi:  1.26E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128337BDBM128337(US8796280, 27)
Affinity DataKi:  1.32E+3nM ΔG°:  -33.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128321BDBM128321(US8796280, 10)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128319BDBM128319(US8796280, 8)
Affinity DataKi:  1.42E+3nM ΔG°:  -33.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128338BDBM128338(US8796280, 28)
Affinity DataKi:  1.47E+3nM ΔG°:  -33.3kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128339BDBM128339(US8796280, 29)
Affinity DataKi:  1.49E+3nM ΔG°:  -33.3kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128315BDBM128315(US8796280, 4)
Affinity DataKi:  1.57E+3nM ΔG°:  -33.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128340BDBM128340(US8796280, 30)
Affinity DataKi:  1.58E+3nM ΔG°:  -33.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128341BDBM128341(US8796280, 31)
Affinity DataKi:  1.59E+3nM ΔG°:  -33.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128342BDBM128342(US8796280, 32)
Affinity DataKi:  1.93E+3nM ΔG°:  -32.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128317BDBM128317(US8796280, 6)
Affinity DataKi:  2.12E+3nM ΔG°:  -32.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128343BDBM128343(US8796280, 33)
Affinity DataKi:  2.21E+3nM ΔG°:  -32.3kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128316BDBM128316(US8796280, 5)
Affinity DataKi:  2.32E+3nM ΔG°:  -32.2kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128318BDBM128318(US8796280, 7)
Affinity DataKi:  2.59E+3nM ΔG°:  -31.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128344BDBM128344(US8796280, 34)
Affinity DataKi:  2.60E+3nM ΔG°:  -31.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128345BDBM128345(US8796280, 35)
Affinity DataKi:  2.64E+3nM ΔG°:  -31.8kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128346BDBM128346(US8796280, 36)
Affinity DataKi:  2.69E+3nM ΔG°:  -31.8kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128347BDBM128347(US8796280, 37)
Affinity DataKi:  2.82E+3nM ΔG°:  -31.7kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128348BDBM128348(US8796280, 38)
Affinity DataKi:  2.90E+3nM ΔG°:  -31.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128349BDBM128349(US8796280, 39)
Affinity DataKi:  2.95E+3nM ΔG°:  -31.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128320BDBM128320(US8796280, 9)
Affinity DataKi:  2.98E+3nM ΔG°:  -31.5kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128350BDBM128350(US8796280, 40)
Affinity DataKi:  3.06E+3nM ΔG°:  -31.5kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128352BDBM128352(US8796280, 42)
Affinity DataKi:  3.90E+3nM ΔG°:  -30.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128351BDBM128351(US8796280, 41)
Affinity DataKi:  3.90E+3nM ΔG°:  -30.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128324BDBM128324(US8796280, 13)
Affinity DataKi:  4.03E+3nM ΔG°:  -30.8kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128353BDBM128353(US8796280, 43)
Affinity DataKi:  4.11E+3nM ΔG°:  -30.7kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128354BDBM128354(US8796280, 44)
Affinity DataKi:  4.44E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128355BDBM128355(US8796280, 45)
Affinity DataKi:  4.51E+3nM ΔG°:  -30.5kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128356BDBM128356(US8796280, 46)
Affinity DataKi:  4.65E+3nM ΔG°:  -30.4kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128322BDBM128322(US8796280, 11)
Affinity DataKi:  5.16E+3nM ΔG°:  -30.2kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128326BDBM128326(US8796280, 15)
Affinity DataKi:  5.38E+3nM ΔG°:  -30.1kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128327BDBM128327(US8796280, 16)
Affinity DataKi:  5.71E+3nM ΔG°:  -29.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128325BDBM128325(US8796280, 14)
Affinity DataKi:  5.85E+3nM ΔG°:  -29.9kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent

TargetProstaglandin D2 receptor 2(Human)
Merck Serono

US Patent
LigandChemical structure of BindingDB Monomer ID 128323BDBM128323(US8796280, 12)
Affinity DataKi:  8.43E+3nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The compounds of the present invention inhibit the binding of PGD2 to its receptor CRTH2. The inhibitory activity can be investigated by a radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2015
Entry Details
US Patent