Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 1177
TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309489BDBM309489(US9603833, Example 111)
Affinity DataIC50: 0.400nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 15581BDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.5nMAssay Description:The compounds of the present invention obtained in the Production Examples were examined for the inhibitory effect on human monoamineoxydase enzymes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309489BDBM309489(US9603833, Example 111)
Affinity DataIC50: 0.5nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309497BDBM309497(US9603833, Example 120)
Affinity DataIC50: 0.600nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309490BDBM309490(US9603833, Example 112)
Affinity DataIC50: 0.700nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309490BDBM309490(US9603833, Example 112)
Affinity DataIC50: 0.700nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309491BDBM309491(US9603833, Example 113)
Affinity DataIC50: 0.700nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309479BDBM309479(US9603833, Example 92)
Affinity DataIC50: 0.800nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309486BDBM309486(US9603833, Example 108)
Affinity DataIC50: 0.800nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309491BDBM309491(US9603833, Example 113)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309476BDBM309476(US9603833, Example 88)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309477BDBM309477(US9603833, Example 89)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309486BDBM309486(US9603833, Example 108)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309474BDBM309474(US9603833, Example 86)
Affinity DataIC50: 1nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309459BDBM309459(US9603833, Example 12)
Affinity DataIC50: 1.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309464BDBM309464(US9603833, Example 45)
Affinity DataIC50: 1.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309492BDBM309492(US9603833, Example 114)
Affinity DataIC50: 1.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309470BDBM309470(US9603833, Example 70)
Affinity DataIC50: 1.30nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309487BDBM309487(US9603833, Example 109)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309475BDBM309475(US9603833, Example 87)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309478BDBM309478(US9603833, Example 90)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309488BDBM309488(US9603833, Example 110)
Affinity DataIC50: 1.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309498BDBM309498(US9603833, Example 121)
Affinity DataIC50: 1.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309473BDBM309473(US9603833, Example 85)
Affinity DataIC50: 1.90nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309492BDBM309492(US9603833, Example 114)
Affinity DataIC50: 2nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309482BDBM309482(US9603833, Example 101)
Affinity DataIC50: 2.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309461BDBM309461(US9603833, Example 30)
Affinity DataIC50: 2.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309498BDBM309498(US9603833, Example 121)
Affinity DataIC50: 2.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309481BDBM309481(US9603833, Example 99)
Affinity DataIC50: 2.5nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309495BDBM309495(US9603833, Example 117)
Affinity DataIC50: 2.70nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309475BDBM309475(US9603833, Example 87)
Affinity DataIC50: 3.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309482BDBM309482(US9603833, Example 101)
Affinity DataIC50: 3.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309480BDBM309480(US9603833, Example 95)
Affinity DataIC50: 3.5nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309488BDBM309488(US9603833, Example 110)
Affinity DataIC50: 3.5nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309465BDBM309465(US9603833, Example 47)
Affinity DataIC50: 3.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309487BDBM309487(US9603833, Example 109)
Affinity DataIC50: 3.70nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309497BDBM309497(US9603833, Example 120)
Affinity DataIC50: 3.70nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309493BDBM309493(US9603833, Example 115)
Affinity DataIC50: 4nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309471BDBM309471(US9603833, Example 74)
Affinity DataIC50: 4.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309496BDBM309496(US9603833, Example 119)
Affinity DataIC50: 4.70nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309500BDBM309500(US9603833, Example 124)
Affinity DataIC50: 4.70nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309460BDBM309460(US9603833, Example 20)
Affinity DataIC50: 5.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309462BDBM309462(US9603833, Example 44)
Affinity DataIC50: 5.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309500BDBM309500(US9603833, Example 124)
Affinity DataIC50: 5.5nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309472BDBM309472(US9603833, Example 83)
Affinity DataIC50: 5.80nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309467BDBM309467(US9603833, Example 59)
Affinity DataIC50: 6.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309480BDBM309480(US9603833, Example 95)
Affinity DataIC50: 6.30nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309499BDBM309499(US9603833, Example 122)
Affinity DataIC50: 6.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309484BDBM309484(US9603833, Example 105)
Affinity DataIC50: 7.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 3(Human)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309484BDBM309484(US9603833, Example 105)
Affinity DataIC50: 7.30nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

Displayed 1 to 50 (of 88 total ) | Next | Last >>
Jump to: