Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 1524
TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329774BDBM329774(US9663523, Example 38 | (−)-(4R)-6-(4-chloro...)
Affinity DataIC50: 20nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329749BDBM329749(US9663523, Example 13 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 30nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329771BDBM329771(US9663523, Example 35 | (−)-6-[(4R)-4-chloro...)
Affinity DataIC50: 30nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329738BDBM329738(US9663523, Example 2 | ethyl (−)-(4R)-[6-(4-...)
Affinity DataIC50: 30nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329775BDBM329775(US9663523, Example 39 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 40nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329776BDBM329776(US9663523, Example 40 | N′-acetyl-2-[(4R)-6-...)
Affinity DataIC50: 40nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329762BDBM329762(US9663523, Example 26 | 1-{[6-(4-chlorophenyl)-1-m...)
Affinity DataIC50: 40nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329751BDBM329751(US9663523, Example 15 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 40nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329773BDBM329773(US9663523, Example 37 | (−)-(4R)-6-(4-Chloro...)
Affinity DataIC50: 50nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329778BDBM329778(US9663523, Example 42 | (+)-(4R)-6-(4-chlorophenyl...)
Affinity DataIC50: 50nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329781BDBM329781(US9663523, Example 45 | (−)-(4R)-6-(4-chloro...)
Affinity DataIC50: 50nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329783BDBM329783(US9663523, Example 47 | 6-(4-chlorophenyl)-8-metho...)
Affinity DataIC50: 50nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329755BDBM329755(US9663523, Example 19 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 50nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329757BDBM329757(US9663523, Example 21 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 80nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329788BDBM329788(US9663523, Example 53 | 2-[(4R)-6-(4-chlorophenyl)...)
Affinity DataIC50: 80nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329766BDBM329766(US9663523, Example 30 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 80nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329782BDBM329782(US9663523, Example 46 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 80nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329772BDBM329772(US9663523, Example 36 | (−)-(4R)-6-(4-chloro...)
Affinity DataIC50: 90nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329790BDBM329790(US9663523, Example 55 | (4R)-6-(4-chlorophenyl)-1-...)
Affinity DataIC50: 90nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329780BDBM329780(US9663523, Example 44 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 90nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329753BDBM329753(US9663523, Example 17 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 90nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329770BDBM329770(US9663523, Example 34 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 90nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329777BDBM329777(US9663523, Example 41 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 100nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329763BDBM329763(US9663523, Example 27 | (−)-1-{[(4R)-6-(4-ch...)
Affinity DataIC50: 110nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329789BDBM329789(US9663523, Example 54 | 6-(4-chlorophenyl)-1-methy...)
Affinity DataIC50: 130nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329740BDBM329740(US9663523, Example 4 | (−)-2-[(4R)-6-(4-chlo...)
Affinity DataIC50: 130nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329779BDBM329779(US9663523, Example 43 | 6-(4-chlorophenyl)-4-[(5-c...)
Affinity DataIC50: 130nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329748BDBM329748(US9663523, Example 12 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 130nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329791BDBM329791(US9663523, Example 56 | 2-{[(4R)-6-(4-chlorophenyl...)
Affinity DataIC50: 180nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329767BDBM329767(US9663523, Example 31 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 180nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329737BDBM329737(US9663523, Example 1 | ethyl [6-(4-chlorophenyl)-1...)
Affinity DataIC50: 180nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329787BDBM329787(US9663523, Example 52 | 2-[(4R)-6-(4-chlorophenyl)...)
Affinity DataIC50: 190nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329745BDBM329745(US9663523, Example 9 | tert-butyl (−)-[(4R)-...)
Affinity DataIC50: 200nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329754BDBM329754(US9663523, Example 18 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 200nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329760BDBM329760(US9663523, Example 24 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 220nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329752BDBM329752(US9663523, Example 16 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 220nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329739BDBM329739(US9663523, Example 3 | 2-[6-(4-chlorophenyl)-1-met...)
Affinity DataIC50: 220nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329786BDBM329786(US9663523, Example 51 | 2-[(4R)-6-(4-chlorophenyl)...)
Affinity DataIC50: 220nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329743BDBM329743(US9663523, Example 7 | ethyl [6-(3-chlorophenyl)-1...)
Affinity DataIC50: 230nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329756BDBM329756(US9663523, Example 20 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 240nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329792BDBM329792(US9663523, Example 57 | (4R)-4-({5-[(benzyloxy)met...)
Affinity DataIC50: 270nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329747BDBM329747(US9663523, Example 11 | (−)-2-[(4R)-6-(3-chl...)
Affinity DataIC50: 300nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329750BDBM329750(US9663523, Example 14 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 310nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329758BDBM329758(US9663523, Example 22 | 3-{[(6-(4-chlorophenyl)-1-...)
Affinity DataIC50: 340nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329784BDBM329784(US9663523, Example 48 | 6-(4-chlorophenyl)-8-(3,5-...)
Affinity DataIC50: 340nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329744BDBM329744(US9663523, Example 8 | tert-butyl [6-(4-chlorophen...)
Affinity DataIC50: 350nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329768BDBM329768(US9663523, Example 32 | 2-[6-(4-chlorophenyl)-1-me...)
Affinity DataIC50: 390nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329759BDBM329759(US9663523, Example 23 | (−)-3-{[(4R)-6-(4-ch...)
Affinity DataIC50: 450nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329769BDBM329769(US9663523, Example 33 | (−)-2-[(4R)-6-(4-chl...)
Affinity DataIC50: 450nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

TargetBromodomain-containing protein 4(Human)
Bayer

US Patent
LigandChemical structure of BindingDB Monomer ID 329742BDBM329742(US9663523, Example 6 | (−)-1 (7-azabicyclo[2...)
Affinity DataIC50: 600nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: