Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 1843
LigandChemical structure of BindingDB Monomer ID 343674BDBM343674(6-Chloro-3-(4-methoxy-1-benzofuran-2-yl)imidazo[1,...)
Affinity DataIC50: 4nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343675BDBM343675(6-Chloro-3-(5-methoxy-1-benzofuran-2-yl)imidazo[1,...)
Affinity DataIC50: 4nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343673BDBM343673(3-(1-Benzofuran-2-yl)-6-[2-(morpholin-2-yl)ethoxy]...)
Affinity DataIC50: 4nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343677BDBM343677(3-(1-Benzofuran-2-yl)-6-{2-[(3R)-morpholin-3-yl]et...)
Affinity DataIC50: 6nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343673BDBM343673(3-(1-Benzofuran-2-yl)-6-[2-(morpholin-2-yl)ethoxy]...)
Affinity DataIC50: 6nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343676BDBM343676(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 7nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343678BDBM343678(3-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 7nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343679BDBM343679(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 8nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343685BDBM343685(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 8nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343682BDBM343682(3-(1-Benzofuran-2-yl)-6-{2-[(3S)-morpholin-3-yl]et...)
Affinity DataIC50: 9nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343698BDBM343698(3-(4-Fluoro-1-benzofuran-2-yl)-6-[(2R)-morpholin-2...)
Affinity DataIC50: 10nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343699BDBM343699(3-(5-Fluoro-1-benzofuran-2-yl)-6-[(2R)-morpholin-2...)
Affinity DataIC50: 10nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343681BDBM343681(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 11nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343700BDBM343700(3-(1-Benzofur-2-yl)-6-chloroimidazo[1,2-b]pyridazi...)
Affinity DataIC50: 11nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343699BDBM343699(3-(5-Fluoro-1-benzofuran-2-yl)-6-[(2R)-morpholin-2...)
Affinity DataIC50: 11nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343680BDBM343680(3-(1-Benzofuran-2-yl)-6-[(2S)-morpholin-2-ylmethox...)
Affinity DataIC50: 12nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343683BDBM343683(3-(1-Benzofuran-2-yl)-6-{2-[(2S)-pyrrolidin-2-yl]e...)
Affinity DataIC50: 12nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343674BDBM343674(6-Chloro-3-(4-methoxy-1-benzofuran-2-yl)imidazo[1,...)
Affinity DataIC50: 12nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343675BDBM343675(6-Chloro-3-(5-methoxy-1-benzofuran-2-yl)imidazo[1,...)
Affinity DataIC50: 13nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343698BDBM343698(3-(4-Fluoro-1-benzofuran-2-yl)-6-[(2R)-morpholin-2...)
Affinity DataIC50: 15nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343688BDBM343688(US9777004, 23 | 3-(1-Benzofuran-2-yl)-6-[(2R)-pyrr...)
Affinity DataIC50: 15nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343684BDBM343684(3-(1-Benzofuran-2-yl)-6-(piperidin-2-ylmethoxy)imi...)
Affinity DataIC50: 16nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343687BDBM343687(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 16nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343701BDBM343701(6-Chloro-3-(5-chloro-1-benzofuran-2-yl)imidazo[1,2...)
Affinity DataIC50: 18nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343676BDBM343676(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 18nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343702BDBM343702(3-(1-Benzofuran-2-yl)-6-[(2R)-morpholin-2-ylmethox...)
Affinity DataIC50: 19nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343678BDBM343678(3-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 20nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343677BDBM343677(3-(1-Benzofuran-2-yl)-6-{2-[(3R)-morpholin-3-yl]et...)
Affinity DataIC50: 20nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343696BDBM343696(3-(1-Benzofuran-2-yl)-6-[(3R)-pyrrolidin-3-yloxy]i...)
Affinity DataIC50: 22nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343679BDBM343679(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 23nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343680BDBM343680(3-(1-Benzofuran-2-yl)-6-[(2S)-morpholin-2-ylmethox...)
Affinity DataIC50: 24nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343686BDBM343686(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 24nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343688BDBM343688(US9777004, 23 | 3-(1-Benzofuran-2-yl)-6-[(2R)-pyrr...)
Affinity DataIC50: 25nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343682BDBM343682(3-(1-Benzofuran-2-yl)-6-{2-[(3S)-morpholin-3-yl]et...)
Affinity DataIC50: 25nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343681BDBM343681(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 25nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343689BDBM343689(3-(1-Benzofuran-2-yl)-6-(piperidin-3-yloxy)imidazo...)
Affinity DataIC50: 25nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343703BDBM343703(6-(Azetidin-3-ylmethoxy)-3-(1-benzofuran-2-yl)imid...)
Affinity DataIC50: 27nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343697BDBM343697(3-(1-Benzofuran-2-yl)-6-[(3R)-piperidin-3-yloxy]im...)
Affinity DataIC50: 28nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343683BDBM343683(3-(1-Benzofuran-2-yl)-6-{2-[(2S)-pyrrolidin-2-yl]e...)
Affinity DataIC50: 30nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343684BDBM343684(3-(1-Benzofuran-2-yl)-6-(piperidin-2-ylmethoxy)imi...)
Affinity DataIC50: 32nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343692BDBM343692(Formic acid-N-(2-{[3-(1-benzofuran-2-yl)imidazo[1,...)
Affinity DataIC50: 36nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343685BDBM343685(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 36nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343686BDBM343686(N-(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazi...)
Affinity DataIC50: 37nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343687BDBM343687(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)
Affinity DataIC50: 38nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343691BDBM343691(3-(5-Chloro-1-benzofuran-2-yl)-6-{2-[(2S)-pyrrolid...)
Affinity DataIC50: 39nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343704BDBM343704(3-(5-Chloro-1-benzofuran-2-yl)-6-[(2R)-morpholin-2...)
Affinity DataIC50: 41nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343688BDBM343688(US9777004, 23 | 3-(1-Benzofuran-2-yl)-6-[(2R)-pyrr...)
Affinity DataIC50: 44nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343696BDBM343696(3-(1-Benzofuran-2-yl)-6-[(3R)-pyrrolidin-3-yloxy]i...)
Affinity DataIC50: 49nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343688BDBM343688(US9777004, 23 | 3-(1-Benzofuran-2-yl)-6-[(2R)-pyrr...)
Affinity DataIC50: 53nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 343697BDBM343697(3-(1-Benzofuran-2-yl)-6-[(3R)-piperidin-3-yloxy]im...)
Affinity DataIC50: 53nMAssay Description:For the assay 50 nL of a 100fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384well microtiter plate (Gr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2019
Entry Details
US Patent

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