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Report error Found 277 Enz. Inhib. hit(s) with all data for entry = 513
TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055925BDBM50055925(CHEMBL3321939 | US9884814, Compound 99)
Affinity DataIC50: 8.60nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275594BDBM275594(US9884814, Compound 196)
Affinity DataIC50: 11nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275605BDBM275605(US9884814, Compound 208)
Affinity DataIC50: 11nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275668BDBM275668(US9884814, Compound 281)
Affinity DataIC50: 13nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275727BDBM275727(US9884814, Compound 341)
Affinity DataIC50: 13nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275512BDBM275512(US9884814, Compound 69)
Affinity DataIC50: 15nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055907BDBM50055907(CHEMBL3321928 | US9884814, Compound 60)
Affinity DataIC50: 17nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275675BDBM275675(US9884814, Compound 288)
Affinity DataIC50: 20nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055892BDBM50055892(CHEMBL3321931 | US9884814, Compound 44)
Affinity DataIC50: 24nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275681BDBM275681(US9884814, Compound 294)
Affinity DataIC50: 24nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275491BDBM275491(US9884814, Compound 46)
Affinity DataIC50: 26nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275488BDBM275488(US9884814, Compound 43)
Affinity DataIC50: 31nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275671BDBM275671(US9884814, Compound 284)
Affinity DataIC50: 35nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275705BDBM275705(US9884814, Compound 319)
Affinity DataIC50: 41nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275619BDBM275619(US9884814, Compound 222)
Affinity DataIC50: 41nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275625BDBM275625(US9884814, Compound 230)
Affinity DataIC50: 42nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275719BDBM275719(US9884814, Compound 333)
Affinity DataIC50: 42nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275624BDBM275624(US9884814, Compound 229)
Affinity DataIC50: 43nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055931BDBM50055931(CHEMBL3321933 | US9884814, Compound 272)
Affinity DataIC50: 44nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275701BDBM275701(US9884814, Compound 315)
Affinity DataIC50: 45nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275725BDBM275725(US9884814, Compound 339)
Affinity DataIC50: 45nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275583BDBM275583(US9884814, Compound 157)
Affinity DataIC50: 46nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275713BDBM275713(US9884814, Compound 327)
Affinity DataIC50: 47nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275696BDBM275696(US9884814, Compound 310)
Affinity DataIC50: 47nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275685BDBM275685(US9884814, Compound 298)
Affinity DataIC50: 48nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275582BDBM275582(US9884814, Compound 156)
Affinity DataIC50: 48nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275587BDBM275587(US9884814, Compound 162)
Affinity DataIC50: 49nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275726BDBM275726(US9884814, Compound 340)
Affinity DataIC50: 49nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275708BDBM275708(US9884814, Compound 322)
Affinity DataIC50: 49nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275471BDBM275471(US9884814, Compound 22)
Affinity DataIC50: 50nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275664BDBM275664(US9884814, Compound 275)
Affinity DataIC50: 51nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275688BDBM275688(US9884814, Compound 301)
Affinity DataIC50: 52nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275549BDBM275549(US9884814, Compound 109)
Affinity DataIC50: 55nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275674BDBM275674(US9884814, Compound 287)
Affinity DataIC50: 56nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275650BDBM275650(US9884814, Compound 261)
Affinity DataIC50: 57nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275533BDBM275533(US9884814, Compound 93)
Affinity DataIC50: 57nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055908BDBM50055908(CHEMBL3321925 | US9884814, Compound 141)
Affinity DataIC50: 58nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275543BDBM275543(US9884814, Compound 103)
Affinity DataIC50: 59nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275673BDBM275673(US9884814, Compound 286)
Affinity DataIC50: 61nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275612BDBM275612(US9884814, Compound 215)
Affinity DataIC50: 63nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275635BDBM275635(US9884814, Compound 243)
Affinity DataIC50: 66nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055934BDBM50055934(CHEMBL3321927 | US9884814, Compound 51)
Affinity DataIC50: 67nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275709BDBM275709(US9884814, Compound 323)
Affinity DataIC50: 67nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275497BDBM275497(US9884814, Compound 53)
Affinity DataIC50: 72nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275599BDBM275599(US9884814, Compound 201)
Affinity DataIC50: 72nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275667BDBM275667(US9884814, Compound 278)
Affinity DataIC50: 74nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275504BDBM275504(US9884814, Compound 61)
Affinity DataIC50: 74nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275498BDBM275498(US9884814, Compound 54)
Affinity DataIC50: 78nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 275672BDBM275672(US9884814, Compound 285)
Affinity DataIC50: 80nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 50055930BDBM50055930(CHEMBL3321934 | US9884814, Compound 276)
Affinity DataIC50: 81nMpH: 5.5 T: 2°CAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details
US Patent

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