Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 2729
TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377141(USRE47351, Compound 19 | (1-{9-[(4S,2R,3R,5R)-3,4-...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377140(USRE47351, Compound 18 | (1-{9-[(4S,2R,3R,5R)-3,4-...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377144(USRE47351, Compound 22 | (1-{9-[(4S,2R,3R,5R)-3,4-...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377143(USRE47351, Compound 21 | (1-{9-[(4S,2R,3R,5R)-3,4-...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377142(USRE47351, Compound 20 | 1-{9-[(4S,2R,3R,5R)-3,4-d...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377134(USRE47351, Compound 12 | Ethyl 1-{9-[(4S,2R,3R,5R)...)
Affinity DataKi:  505nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377139(USRE47351, Compound 17 | 1-{9-[(4S,2R,3R,5R)-3,4-d...)
Affinity DataKi: >1.00E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM50152084(1-[6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-tetrah...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377137(USRE47351, Compound 15 | (4S,2R,3R,5R)-2-{6-Amino2...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377136(USRE47351, Compound 14 | (4S,2R,3R,5R)-2-{6-Amino-...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAdenosine receptor A2a(Guinea pig)
Gilead Sciences

US Patent
LigandPNGBDBM377135(USRE47351, Compound 13 | (4S,2R,3R,5R)-2-{6-Amino-...)
Affinity DataKi:  5.50E+3nMAssay Description:Compounds of this invention were assayed to determine their affinity for the A2A receptor in a pig striatum membrane prep. Briefly, 0.2 mg of pig str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent