Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 11024
TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM586110(USRE49340, Rank 1 | 5-O-Desmethyl- Omeprazole (RS-...)
Affinity DataIC50: 1.19E+3nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)
Affinity DataIC50: 3.28E+3nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM586207(USRE49340, Rank 3 | PM-BRL 36610A)
Affinity DataIC50: 3.45E+3nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM586222(USRE49340, Rank 4 | PM-BRL 36583A)
Affinity DataIC50: 3.67E+3nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM84745(DULOXETINE | LY-248686 | CAS_136434-34-9 | LY24868...)
Affinity DataIC50: 5.47E+3nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM586429(Amodiaquin | USRE49340, Rank 6 | BDBM50041457)
Affinity DataIC50: 9.76E+4nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM50122054(N-desmethyl-Clozapine | 8-Chloro-11-piperazin-1-yl...)
Affinity DataIC50: 1.02E+5nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM586486(USRE49340, Rank 8 | Esomeprazole)
Affinity DataIC50: 1.06E+5nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent

TargetD-amino-acid oxidase(Human)
National Taiwan University

US Patent
LigandPNGBDBM50105085(US9233167, Nalbuphine | 17-cyclobutylmethyl-4,5alp...)
Affinity DataIC50: 1.21E+5nMAssay Description:The DAAO enzymatic activity assay was modified according to the report of Oguri et al (Oguri, S., Screening of d-amino acid oxidase inhibitor by a ne...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
US Patent