Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50036733
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369433(CHEMBL1202108)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369433(CHEMBL1202108)
Affinity DataKi:  0.0450nMAssay Description:The binding affinity towards thrombin obtained from human purified enzymes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079215([3-(3-Carbamimidoyl-phenyl)-5-(2'-methanesulfonyl-...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079216([3-(3-Carbamimidoyl-phenyl)-5-(3-fluoro-2'-sulfamo...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  7nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  7nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079220([3-(3-Carbamimidoyl-phenyl)-5-(3-methyl-2'-sulfamo...)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079222({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  12nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079222({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  12nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079222({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  12nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079222({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  12nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  17nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  17nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079219({3-(3-Carbamimidoyl-phenyl)-5-[6-(2-sulfamoyl-phen...)
Affinity DataKi:  19nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079210([3-(3-Carbamimidoyl-phenyl)-5-(2'-trifluoromethyl-...)
Affinity DataKi:  28nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079217(4'-{[3-(3-Carbamimidoyl-phenyl)-5-methoxycarbonylm...)
Affinity DataKi:  53nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369433(CHEMBL1202108)
Affinity DataKi:  55nMAssay Description:The binding affinity was measured on trypsin obtained from Human purified enzymesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079225([3-(3-Carbamimidoyl-phenyl)-5-(2'-methoxy-biphenyl...)
Affinity DataKi:  62nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079212([3-(3-Carbamimidoyl-phenyl)-5-(2'-methylsulfanyl-b...)
Affinity DataKi:  66nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079223([3-(3-Carbamimidoyl-phenyl)-5-(3'-sulfamoyl-biphen...)
Affinity DataKi:  68nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  98nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  98nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  98nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079215([3-(3-Carbamimidoyl-phenyl)-5-(2'-methanesulfonyl-...)
Affinity DataKi:  100nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079216([3-(3-Carbamimidoyl-phenyl)-5-(3-fluoro-2'-sulfamo...)
Affinity DataKi:  120nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072445(CHEMBL139063 | CHEMBL279628 | [3-(3-Carbamimidoyl-...)
Affinity DataKi:  121nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  130nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079211({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  130nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079219({3-(3-Carbamimidoyl-phenyl)-5-[6-(2-sulfamoyl-phen...)
Affinity DataKi:  180nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079227([3-(3-Carbamimidoyl-phenyl)-5-(3'-methoxy-biphenyl...)
Affinity DataKi:  200nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079214([3-(3-Carbamimidoyl-phenyl)-5-(2'-methyl-biphenyl-...)
Affinity DataKi:  210nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079224([5-(Biphenyl-4-ylcarbamoyl)-3-(3-carbamimidoyl-phe...)
Affinity DataKi:  220nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079210([3-(3-Carbamimidoyl-phenyl)-5-(2'-trifluoromethyl-...)
Affinity DataKi:  230nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079226([3-(3-Carbamimidoyl-phenyl)-5-(3'-trifluoromethyl-...)
Affinity DataKi:  240nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079221([3-(3-Carbamimidoyl-phenyl)-5-(3'-methyl-biphenyl-...)
Affinity DataKi:  240nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079212([3-(3-Carbamimidoyl-phenyl)-5-(2'-methylsulfanyl-b...)
Affinity DataKi:  260nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079220([3-(3-Carbamimidoyl-phenyl)-5-(3-methyl-2'-sulfamo...)
Affinity DataKi:  300nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079217(4'-{[3-(3-Carbamimidoyl-phenyl)-5-methoxycarbonylm...)
Affinity DataKi:  300nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079225([3-(3-Carbamimidoyl-phenyl)-5-(2'-methoxy-biphenyl...)
Affinity DataKi:  310nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079222({3-(3-Carbamimidoyl-phenyl)-5-[5-(2-sulfamoyl-phen...)
Affinity DataKi:  330nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079223([3-(3-Carbamimidoyl-phenyl)-5-(3'-sulfamoyl-biphen...)
Affinity DataKi:  340nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079214([3-(3-Carbamimidoyl-phenyl)-5-(2'-methyl-biphenyl-...)
Affinity DataKi:  390nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079227([3-(3-Carbamimidoyl-phenyl)-5-(3'-methoxy-biphenyl...)
Affinity DataKi:  390nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
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