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Found 13 Enz. Inhib. hit(s) with all data for entry = 50009348
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  43nMAssay Description:Inhibition of monoamine [3H]-DA reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  43nMAssay Description:Inhibition of monoamine [3H]-DA reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082393(CHEMBL441075 | piperidine based analogue of cocain...)
Affinity DataKi:  96nMAssay Description:Binding affinity against dopamine transporter (DAT) was evaluated using competitive binding assay and [3H]-mazindol as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  110nMAssay Description:Inhibition of monoamine [3H]-DA reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  112nMAssay Description:Binding affinity against dopamine transporter (DAT) was evaluated using competitive binding assay and [3H]-mazindol as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082393(CHEMBL441075 | piperidine based analogue of cocain...)
Affinity DataKi:  193nMAssay Description:Norepinephrine transporter activity was determined by inhibition of monoamine [3H]-NE reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082393(CHEMBL441075 | piperidine based analogue of cocain...)
Affinity DataKi:  231nMAssay Description:Norepinephrine transporter activity was determined by inhibition of monoamine [3H]-NE reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082393(CHEMBL441075 | piperidine based analogue of cocain...)
Affinity DataKi:  243nMAssay Description:Inhibition of monoamine [3H]-5-HT reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  888nMAssay Description:Inhibition of monoamine [3H]-5-HT reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  888nMAssay Description:Inhibition of monoamine [3H]-5-HT reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  2.03E+3nMAssay Description:Norepinephrine transporter activity was determined by inhibition of monoamine [3H]-NE reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082392(CHEMBL324631 | PIPERIDINE BASED ANALOGUE OF COCAIN...)
Affinity DataKi:  2.03E+3nMAssay Description:Norepinephrine transporter activity was determined by inhibition of monoamine [3H]-NE reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50082395((3S,4S)-4-(4-Chloro-phenyl)-1-methyl-3-propyl-pipe...)
Affinity DataIC50:  3nMAssay Description:Binding affinity towards dopamine transporter (DAT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed