Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50036899
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084878(Butyl-[8-(2,4-dichloro-phenyl)-2,7-dimethyl-pyrazo...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084876([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084880(Cyclopropylmethyl-[8-(2,4-dichloro-phenyl)-2,7-dim...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084873([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084877([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084869([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084881([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084874(Butyl-[2,5-dimethyl-7-(2,4,6-trimethyl-phenyl)-7H-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084870([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084875(DMP696 | [8-(2,4-dichloro-phenyl)-2,7-dimethyl-pyr...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084879([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084872([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084868([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50084871([8-(2,4-Dichloro-phenyl)-2,7-dimethyl-pyrazolo[1,5...)
Affinity DataKi:  44.5nMAssay Description:Displacement of [125I]-tyrosine-ovine-CRF from human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed