Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for entry = 50036822
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089779(4-cyclopropylmethyl-14-(3,4-diformylphenylcarboxam...)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]- diprenorphine binding to Opioid receptor mu 1 (83 fmol/mg protein) stably expressed in membranes from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089779(4-cyclopropylmethyl-14-(3,4-diformylphenylcarboxam...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]diprenorphine binding to Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089779(4-cyclopropylmethyl-14-(3,4-diformylphenylcarboxam...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of [3H]- diprenorphine binding to Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed