Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50010236
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092301(1-(Benzo[b]thiophene-2-carbonyl)-piperidine-4-carb...)
Affinity DataKi:  9nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataKi:  15nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataKi:  25nMAssay Description:Inhibition of human Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092297(1-(Naphthalene-2-carbonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  30nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092294(1-(Quinoline-6-carbonyl)-piperidine-4-carboxylic a...)
Affinity DataKi:  160nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092298(1-(Naphthalene-2-sulfonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  450nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092300(1-[(E)-(3-Phenyl-acryloyl)]-piperidine-4-carboxyli...)
Affinity DataKi:  460nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092295(1-Benzoyl-piperidine-4-carboxylic acid (1-benzyl-2...)
Affinity DataKi:  560nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092299(1-(Quinoline-3-carbonyl)-piperidine-4-carboxylic a...)
Affinity DataKi:  670nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092302(1-(Naphthalene-2-sulfonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  810nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092305(1-(Naphthalene-2-carbonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  960nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092303(1-[(E)-(3-Phenyl-acryloyl)]-piperidine-4-carboxyli...)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092301(1-(Benzo[b]thiophene-2-carbonyl)-piperidine-4-carb...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092297(1-(Naphthalene-2-carbonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  7.30E+3nMAssay Description:Inhibition of human Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092304(1-((E)-3-Pyridin-4-yl-acryloyl)-piperidine-4-carbo...)
Affinity DataKi:  1.35E+4nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092307(1-Naphthalen-2-ylmethyl-piperidine-4-carboxylic ac...)
Affinity DataKi:  1.36E+4nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092306(1-[(E)-(3-Phenyl-acryloyl)]-piperidine-4-carboxyli...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Knoll

Curated by ChEMBL
LigandPNGBDBM50092296(1-(Naphthalene-2-sulfonyl)-piperidine-4-carboxylic...)
Affinity DataKi:  8.00E+5nMAssay Description:Inhibition of Suc-Leu-Tyr-AMC binding to human mu-calpain from erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed