Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50010260
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092516(3-{[(Methoxycarbonyl-pyridin-2-yl-methyl)-methyl-a...)
Affinity DataKi:  15nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092518(3-[{[Methoxycarbonyl-(4-methoxy-phenyl)-methyl]-me...)
Affinity DataKi:  18nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092515(3-((3-Hydroxy-phenyl)-{[(3-hydroxy-phenyl)-methoxy...)
Affinity DataKi:  20nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092521(3-((3-Fluoro-phenyl)-{[(3-fluoro-phenyl)-methoxyca...)
Affinity DataKi:  26nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092520(3-((4-Fluoro-phenyl)-{[(4-fluoro-phenyl)-methoxyca...)
Affinity DataKi:  140nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092519(3-{[(Methoxycarbonyl-quinolin-2-yl-methyl)-methyl-...)
Affinity DataKi:  190nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092517(3-{[(Carboxy-phenyl-methyl)-methyl-amino]-phenyl-m...)
Affinity DataKi:  210nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092514(3-{[(Methoxycarbonyl-m-tolyl-methyl)-methyl-amino]...)
Affinity DataKi:  820nMAssay Description:Inhibition against [3H]-CI 977 rat Opioid receptor kappa 1 at 10 micromol/LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of WüRzburg

Curated by ChEMBL
LigandPNGBDBM50092513(3-((4-Chloro-phenyl)-{[(4-chloro-phenyl)-ethoxycar...)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibition against [3H]-diprenorphine human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed