Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 615
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4522BDBM4522(4-[(2,4-dichlorophenyl)amino]-7-[3-(4-hydroxypiper...)
Affinity DataIC50: 3.5nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4520BDBM4520(4-Phenylamino-3-quinolinecarbonitrile deriv. 2a | ...)
Affinity DataIC50: 3.80nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4515BDBM4515(4-[(4-Chloro-2-iodophenyl)amino]-6,7-dimethoxy-3-q...)
Affinity DataIC50: 6.20nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4521BDBM4521(4-[(2,4-dichlorophenyl)amino]-6-methoxy-7-[3-(4-me...)
Affinity DataIC50: 8.70nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4514BDBM4514(4-[(2-bromo-4-chlorophenyl)amino]-6,7-dimethoxyqui...)
Affinity DataIC50: 10nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4504BDBM4504(4-[(2,4-Dichlorophenyl)amino]-6,7-diethoxyquinolin...)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4517BDBM4517(4-[(4-bromo-2-chlorophenyl)amino]-6,7-dimethoxyqui...)
Affinity DataIC50: 15nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4518BDBM4518(4-[(2,4-Dichlorophenyl)amino]-6,7-bis(3-morpholin-...)
Affinity DataIC50: 19nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4492BDBM4492(CHEMBL101917 | 4-[(2,4-dichlorophenyl)amino]-6,7-d...)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4509BDBM4509(4-[(2,5-Dichlorophenyl)amino]-6,7-dimethoxy-3-quin...)
Affinity DataIC50: 40nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4507BDBM4507(4-[(4-Chlorophenyl)amino]-6,7-dimethoxy-3-quinolin...)
Affinity DataIC50: 53nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4457BDBM4457(4-Phenylamino-3-quinolinecarbonitrile deriv. 2r | ...)
Affinity DataIC50: 53nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4512BDBM4512(4-[(3,4-Dichlorophenyl)amino]-6,7-dimethoxy-3-quin...)
Affinity DataIC50: 57nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4510BDBM4510(4-[(2,6-dichlorophenyl)amino]-6,7-dimethoxyquinoli...)
Affinity DataIC50: 61nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4494BDBM4494(quinazoline deriv. 4a | (2,4-Dichlorophenyl)(6,7-d...)
Affinity DataIC50: 84nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4508BDBM4508(4-[(2,3-Dichlorophenyl)amino]-6,7-dimethoxy-3-quin...)
Affinity DataIC50: 90nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4506BDBM4506(4-[(2-chlorophenyl)amino]-6,7-dimethoxyquinoline-3...)
Affinity DataIC50: 95nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4516BDBM4516(4-[(2-Chloro-4-iodophenyl)amino]-6,7-dimethoxy-3-q...)
Affinity DataIC50: 95nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4505BDBM4505(4-[(2,4-Dichlorophenyl)amino]-6,7-di-n-butoxy-3-qu...)
Affinity DataIC50: 160nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4502BDBM4502(4-[(2,4-Dichlorophenyl)amino]-7-methoxy-3-quinolin...)
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4519BDBM4519(4-[(2,4-dichlorophenyl)amino]-7-methoxy-6-[3-(morp...)
Affinity DataIC50: 220nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4493BDBM4493(4-[(2,4-Dichlorophenyl)amino]-6,7-dimethoxyquinazo...)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4499BDBM4499(4-[(2,4-Dichlorophenyl)amino]-6,7-dimethoxy-3-quin...)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4501BDBM4501(4-[(2,4-dichlorophenyl)amino]-6-methoxyquinoline-3...)
Affinity DataIC50: 320nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4511BDBM4511(4-[(3,5-dichlorophenyl)amino]-6,7-dimethoxyquinoli...)
Affinity DataIC50: 1.10E+3nMAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4500BDBM4500(4-[(2,4-dichlorophenyl)amino]-5-methoxyquinoline-3...)
Affinity DataIC50: 1.20E+3nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4496BDBM4496(4-[(2,4-dichlorophenyl)sulfanyl]-6,7-dimethoxyquin...)
Affinity DataIC50: 2.20E+3nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4503BDBM4503(4-[(2,4-dichlorophenyl)amino]-5,7-dimethoxyquinoli...)
Affinity DatapH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4495BDBM4495(4-(2,4-dichlorophenoxy)-6,7-dimethoxyquinoline-3-c...)
Affinity DatapH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4497BDBM4497(4-{[(2,4-dichlorophenyl)methyl]amino}-6,7-dimethox...)
Affinity DatapH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth-Ayerst Research

LigandChemical structure of BindingDB Monomer ID 4498BDBM4498(4-(2,4-Dichlorophenylmethylamino)-6,7-dimethoxy-3-...)
Affinity DatapH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2005
Entry Details Article
PubMed