Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50010705
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  1nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097809((S)-2-[(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmet...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097817((S)-2-({5-[(3-Cyclohexylmethyl-3H-imidazol-4-ylmet...)
Affinity DataIC50:  41nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097813(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50:  220nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097810((S)-2-({5-[(3-Biphenyl-4-ylmethyl-3H-imidazol-4-yl...)
Affinity DataIC50:  260nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097811(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50:  380nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097812(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50:  640nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097815((S)-2-({5-[(1-Cyclohexylmethyl-1H-imidazol-4-ylmet...)
Affinity DataIC50:  780nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097808((S)-4-Methylsulfanyl-2-({5-[(1-naphthalen-1-ylmeth...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097816(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097809((S)-2-[(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmet...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097818((S)-2-({5-[(1-Biphenyl-4-ylmethyl-1H-imidazol-4-yl...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097813(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097814((S)-2-[(5-{[(1H-Imidazol-4-ylmethyl)-amino]-methyl...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of mammalian FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097816(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097811(5-{[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-ami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097818((S)-2-({5-[(1-Biphenyl-4-ylmethyl-1H-imidazol-4-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097810((S)-2-({5-[(3-Biphenyl-4-ylmethyl-3H-imidazol-4-yl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50097808((S)-4-Methylsulfanyl-2-({5-[(1-naphthalen-1-ylmeth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian H-Ras processing in NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed