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Found 16 Enz. Inhib. hit(s) with all data for entry = 50010728
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50:  220nMAssay Description:Inhibitition of binding of [3H]-spiroperidol to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50:  430nMAssay Description:Inhibitition of binding of [3H]-SCH-23,390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50:  450nMAssay Description:Inhibitition of binding of [3H]-SCH-23,390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50028970(6-Amino-5,6,7,8-tetrahydro-naphthalene-1,2-diol | ...)
Affinity DataIC50:  700nMAssay Description:Inhibitition of binding of [3H]-spiroperidol to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitition of binding of [3H]-SCH-23,390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50219332(CHEMBL133432)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219332(CHEMBL133432)
Affinity DataIC50:  6.75E+4nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219331(1,2,3,4,4A,5,10,10A-Octahydro-Benzo[G]Quinoline | ...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50:  6.67E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Crete

Curated by ChEMBL
LigandPNGBDBM50098074(1-Benzyl-6-methoxy-1,2,3,4,4a,5,10,10a-octahydro-b...)
Affinity DataIC50:  6.67E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed