Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50011096
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM17659((R,S)-2-phosphonomethylpentanedioic acid | 2-(phos...)
Affinity DataIC50:  5.10nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102256(2-[3-(1-Carboxy-2-mercapto-ethyl)-ureido]-pentaned...)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102259(2-[(2,4-Dicarboxy-butyl)-hydroxy-phosphinoylmethyl...)
Affinity DataIC50:  21.7nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102255(2-[3-(2-tert-Butylsulfanyl-1-carboxy-ethyl)-ureido...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102257(2-[3-(1,2-Dicarboxy-ethyl)-ureido]-pentanedioic ac...)
Affinity DataIC50:  46.1nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase IIusing a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102258((S)-2-[3-((S)-3-Carboxy-1-carboxy-propyl)-ureido]-...)
Affinity DataIC50:  47nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102260(2-(2-Amino-4-carboxy-butyrylamino)-pentanedioic ac...)
Affinity DataIC50:  750nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase II, using a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102262(2-(2-Amino-3-carboxy-propionylamino)-pentanedioic ...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase IIusing a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102261(2-[3-(1,2-Dicarboxy-ethyl)-ureido]-succinic acid |...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory activity of the compound against expressed rat Glutamate carboxypeptidase IIusing a substrate concentration of 5 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed