Affinity DataIC50: 3.20nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 3.89E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 4.68E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13E+3nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1A-adrenoreceptors on isolated prostatic Vas deferens from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 4.17E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair
Affinity DataIC50: 6.76E+4nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1B-adrenoreceptors on isolated spleen from ratMore data for this Ligand-Target Pair