Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50011264
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104334(1-(2-Chloro-2-phenyl-ethyl)-4-phenethylamino-1H-py...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104330(1-(2-Chloro-2-phenyl-ethyl)-4-pyrrolidin-1-yl-1H-p...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104335(1-(2-Chloro-2-phenyl-ethyl)-4-propylamino-1H-pyraz...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104339(1-(2-Chloro-2-phenyl-ethyl)-4-cyclopropylamino-1H-...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104337(4-Benzylamino-1-(2-chloro-2-phenyl-ethyl)-1H-pyraz...)
Affinity DataKi:  139nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104340(1-(2-Chloro-2-phenyl-ethyl)-4-(2-ethoxy-ethylamino...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104336(1-(2-Chloro-2-phenyl-ethyl)-4-phenylamino-1H-pyraz...)
Affinity DataKi:  348nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104331(1-(2-Chloro-2-phenyl-ethyl)-4-morpholin-4-yl-1H-py...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104338(1-(2-Chloro-2-phenyl-ethyl)-4-(4-methyl-piperazin-...)
Affinity DataKi:  2.14E+3nMAssay Description:Displacement of [3H]-CGS-21,680 binding at A2A adenosine receptor in bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104332(4-Butylamino-1-(2-chloro-2-phenyl-ethyl)-1H-pyrazo...)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Facoltà

Curated by ChEMBL
LigandPNGBDBM50104333(4-tert-Butylamino-1-(2-chloro-2-phenyl-ethyl)-1H-p...)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor in bovine cortical membrane expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed