Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50011357
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105701BDBM50105701(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-...)
Affinity DataIC50: 33nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105698BDBM50105698(2-(3-Benzyl-2-imino-2,3-dihydro-benzoimidazol-1-yl...)
Affinity DataIC50: 65nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105697BDBM50105697(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-...)
Affinity DataIC50: 98nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105702BDBM50105702(2-(3-Butyl-2-imino-2,3-dihydro-benzoimidazol-1-yl)...)
Affinity DataIC50: 359nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105700BDBM50105700(2-[3-(4-tert-Butyl-benzyl)-2-imino-2,3-dihydro-ben...)
Affinity DataIC50: 734nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105706BDBM50105706(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(2-imino-...)
Affinity DataIC50: 900nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105703BDBM50105703(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(3-heptyl...)
Affinity DataIC50: 964nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105699BDBM50105699(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[3-(3,4-d...)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105705BDBM50105705(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-(2-imino-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105704BDBM50105704(1-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-2-[2-imino-...)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibitory concentration against potent thrombin receptor-1 (PAR-1) on human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed