Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50011398
LigandPNGBDBM50067584(2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bipheny...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16182((2S)-2-[(4-{[(1H-imidazol-4-ylmethyl)amino]methyl}...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106110([1-(3-Methyl-3H-imidazol-4-ylmethyl)-4-naphthalen-...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106112([1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-1-yl-1H-p...)
Affinity DataIC50: 16nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106113((4-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106111([1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-1-yl-1H-p...)
Affinity DataIC50: 65nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106114((2-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50: 88nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106117([1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-1-yl-1H-p...)
Affinity DataIC50: 115nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106116((3-Bromo-phenyl)-[1-(3H-imidazol-4-ylmethyl)-4-nap...)
Affinity DataIC50: 150nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106118([4-Anthracen-9-yl-1-(3H-imidazol-4-ylmethyl)-1H-py...)
Affinity DataIC50: 470nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106120([1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-1-yl-1H-p...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106119([1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-2-yl-1H-p...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50106115([1-(3H-Imidazol-4-ylmethyl)-4-phenyl-1H-pyrrol-3-y...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of [3H]FPP incorporation into Ha-ras protein by FarnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed