Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50011487
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107034BDBM50107034(N-(4-Butoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 560nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107034BDBM50107034(N-(4-Butoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 630nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107029BDBM50107029(N-(4-Ethoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 760nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107043BDBM50107043(N-(4-Methoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidin...)
Affinity DataIC50: 820nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107032BDBM50107032(N-(Naphthalene-1-carbonyl)-N'-(4-phenyl-butyl)-gua...)
Affinity DataIC50: 860nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107029BDBM50107029(N-(4-Ethoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107031BDBM50107031(N-(4-Methyl-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107030BDBM50107030(N-(2-Methyl-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107046BDBM50107046(N-(4-Phenyl-butyl)-N'-(3,4,5-trimethoxy-benzoyl)-g...)
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107039BDBM50107039(N-(2,3-Dichloro-benzoyl)-N'-(4-phenyl-butyl)-guani...)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107046BDBM50107046(N-(4-Phenyl-butyl)-N'-(3,4,5-trimethoxy-benzoyl)-g...)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107030BDBM50107030(N-(2-Methyl-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107045BDBM50107045(N-[2-(5-Methoxy-1H-indol-3-yl)-ethyl]-N'-(4-methyl...)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107045BDBM50107045(N-[2-(5-Methoxy-1H-indol-3-yl)-ethyl]-N'-(4-methyl...)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107020BDBM50107020(N-(4-Methyl-benzoyl)-N'-(3,4,5-trimethoxy-phenyl)-...)
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107050BDBM50107050(N-(4-Isopropyl-phenyl)-N'-(4-methyl-benzoyl)-guani...)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107035BDBM50107035(N-[2-(4-Chloro-phenyl)-ethyl]-N'-(4-methyl-benzoyl...)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107025BDBM50107025(N-(4-Isopropoxy-phenyl)-N'-(4-methyl-benzoyl)-guan...)
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107043BDBM50107043(N-(4-Methoxy-benzoyl)-N'-(4-phenyl-butyl)-guanidin...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107037BDBM50107037(N-(4-Methyl-benzoyl)-N'-(5-phenyl-pentyl)-guanidin...)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107038BDBM50107038(N-(4-Phenyl-butyl)-N'-(thiophene-2-carbonyl)-guani...)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107051BDBM50107051(N-(4-Methyl-benzoyl)-N'-naphthalen-1-ylmethyl-guan...)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107044BDBM50107044(N-(4-Methyl-benzoyl)-N'-phenethyl-guanidine | CHEM...)
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107017BDBM50107017(N-(4-Methyl-benzoyl)-N'-(3-phenoxy-propyl)-guanidi...)
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107039BDBM50107039(N-(2,3-Dichloro-benzoyl)-N'-(4-phenyl-butyl)-guani...)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107031BDBM50107031(N-(4-Methyl-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107021BDBM50107021(N-(4-Methyl-benzoyl)-N'-(2-phenoxy-ethyl)-guanidin...)
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107052BDBM50107052(N-(2,5-Dichloro-benzoyl)-N'-(4-phenyl-butyl)-guani...)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107048BDBM50107048(N-(4-Methyl-benzoyl)-N'-naphthalen-1-yl-guanidine ...)
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107027BDBM50107027(N-[2-(4-Methoxy-1H-indol-3-yl)-ethyl]-N'-(4-methyl...)
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107037BDBM50107037(N-(4-Methyl-benzoyl)-N'-(5-phenyl-pentyl)-guanidin...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107036BDBM50107036(N-(4-Chloro-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107057BDBM50107057(N-Benzyl-N'-(4-methyl-benzoyl)-guanidine | CHEMBL1...)
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107023BDBM50107023(N-(2-Benzylsulfanyl-ethyl)-N'-(4-methyl-benzoyl)-g...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107027BDBM50107027(N-[2-(4-Methoxy-1H-indol-3-yl)-ethyl]-N'-(4-methyl...)
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107032BDBM50107032(N-(Naphthalene-1-carbonyl)-N'-(4-phenyl-butyl)-gua...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107049BDBM50107049(N-Methyl-N'-(4-methyl-benzoyl)-N''-(4-phenyl-butyl...)
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107036BDBM50107036(N-(4-Chloro-benzoyl)-N'-(4-phenyl-butyl)-guanidine...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107038BDBM50107038(N-(4-Phenyl-butyl)-N'-(thiophene-2-carbonyl)-guani...)
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107053BDBM50107053(N-(2-Isopropyl-phenyl)-N'-(4-methyl-benzoyl)-guani...)
Affinity DataIC50: 4.36E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107053BDBM50107053(N-(2-Isopropyl-phenyl)-N'-(4-methyl-benzoyl)-guani...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107018BDBM50107018(N-(4-Methyl-benzoyl)-N'-(2-thiophen-2-yl-ethyl)-gu...)
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107040BDBM50107040(N-(2,6-Dichloro-benzoyl)-N'-(4-phenyl-butyl)-guani...)
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107026BDBM50107026(N-(4-Methyl-benzoyl)-N'-(3-phenyl-propyl)-guanidin...)
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107040BDBM50107040(N-(2,6-Dichloro-benzoyl)-N'-(4-phenyl-butyl)-guani...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107054BDBM50107054(N-((1E)-amino{methyl[(3-methylphenyl)thio]amino}me...)
Affinity DataIC50: 5.44E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107017BDBM50107017(N-(4-Methyl-benzoyl)-N'-(3-phenoxy-propyl)-guanidi...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107044BDBM50107044(N-(4-Methyl-benzoyl)-N'-phenethyl-guanidine | CHEM...)
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107025BDBM50107025(N-(4-Isopropoxy-phenyl)-N'-(4-methyl-benzoyl)-guan...)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Cenes Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50107026BDBM50107026(N-(4-Methyl-benzoyl)-N'-(3-phenyl-propyl)-guanidin...)
Affinity DataIC50: 6.03E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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