Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50037073
LigandPNGBDBM50108781(2-{[1-(2-Amino-3-mercapto-propionyl)-piperidin-4-y...)
Affinity DataIC50: 20nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108780(2-{2-[4-(2-Amino-3-methylsulfanyl-propylamino)-3-m...)
Affinity DataIC50: 34nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50048955(2-[4-(2-Amino-3-mercapto-propionylamino)-benzoylam...)
Affinity DataIC50: 72nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108780(2-{2-[4-(2-Amino-3-methylsulfanyl-propylamino)-3-m...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108784(2-{Benzoyl-[1-(1H-imidazol-4-ylmethyl)-piperidin-4...)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108785(2-[Benzoyl-(1-thiazol-4-ylmethyl-piperidin-4-yl)-a...)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108783(2-{Benzoyl-[1-(thiazole-4-carbonyl)-piperidin-4-yl...)
Affinity DataIC50: 5.25E+4nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108784(2-{Benzoyl-[1-(1H-imidazol-4-ylmethyl)-piperidin-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108781(2-{[1-(2-Amino-3-mercapto-propionyl)-piperidin-4-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108783(2-{Benzoyl-[1-(thiazole-4-carbonyl)-piperidin-4-yl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50048955(2-[4-(2-Amino-3-mercapto-propionylamino)-benzoylam...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108785(2-[Benzoyl-(1-thiazol-4-ylmethyl-piperidin-4-yl)-a...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50409604(CHEMBL2094059)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Geranylgeranyl transferase type I (GGPT I) catalyzed transfer of GGPP to dansyl-GCVLLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50108786(2-(Benzoyl-piperidin-4-yl-amino)-4-methylsulfanyl-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Farnesyltransferase catalyzed transfer of the FPP moiety to dansyl-GCVLSMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed