Compile Data Set for Download or QSAR
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Found 34 Enz. Inhib. hit(s) with all data for entry = 50011716
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109666(4'-Pyrimidin-2-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50091105(4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109667(4'-Pyridin-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109670(4'-Pyridin-3-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109659(4'-[1,3,4]Oxadiazol-2-yl-biphenyl-2-sulfonic acid ...)
Affinity DataKi:  4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109668(4'-Thiazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109664(4'-Pyrazin-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109663(4'-Pyrazol-1-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109672(4'-(1-Methyl-1H-imidazol-2-yl)-biphenyl-2-sulfonic...)
Affinity DataKi:  19nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109660(4'-Pyrimidin-4-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  25nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109662(4'-(1-Oxy-pyridin-2-yl)-biphenyl-2-sulfonic acid (...)
Affinity DataKi:  37nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109673(CHEMBL149763 | [1,1';4',1'']Terphenyl-2-sulfonic a...)
Affinity DataKi:  38nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109661(4'-(1H-Imidazol-2-yl)-biphenyl-2-sulfonic acid (3,...)
Affinity DataKi:  44nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109671(4'-(4,6-Dimethoxy-pyrimidin-2-yl)-biphenyl-2-sulfo...)
Affinity DataKi:  220nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109674(4'-Isoxazol-5-yl-biphenyl-2-sulfonic acid (3,4-dim...)
Affinity DataKi:  270nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109665(4'-Pyrimidin-5-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  300nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109669(4'-(1H-Tetrazol-5-yl)-biphenyl-2-sulfonic acid (3,...)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109667(4'-Pyridin-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109663(4'-Pyrazol-1-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  9.40E+3nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109666(4'-Pyrimidin-2-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  1.60E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50091105(4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  1.87E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109673(CHEMBL149763 | [1,1';4',1'']Terphenyl-2-sulfonic a...)
Affinity DataKi:  2.00E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109670(4'-Pyridin-3-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  2.00E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109664(4'-Pyrazin-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  2.20E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109662(4'-(1-Oxy-pyridin-2-yl)-biphenyl-2-sulfonic acid (...)
Affinity DataKi:  3.08E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109674(4'-Isoxazol-5-yl-biphenyl-2-sulfonic acid (3,4-dim...)
Affinity DataKi:  3.90E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109671(4'-(4,6-Dimethoxy-pyrimidin-2-yl)-biphenyl-2-sulfo...)
Affinity DataKi:  4.80E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109668(4'-Thiazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...)
Affinity DataKi:  5.20E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109659(4'-[1,3,4]Oxadiazol-2-yl-biphenyl-2-sulfonic acid ...)
Affinity DataKi:  7.50E+4nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109672(4'-(1-Methyl-1H-imidazol-2-yl)-biphenyl-2-sulfonic...)
Affinity DataKi:  1.20E+5nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109660(4'-Pyrimidin-4-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  1.30E+5nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109661(4'-(1H-Imidazol-2-yl)-biphenyl-2-sulfonic acid (3,...)
Affinity DataKi:  1.50E+5nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109665(4'-Pyrimidin-5-yl-biphenyl-2-sulfonic acid (3,4-di...)
Affinity DataKi:  1.70E+5nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50109669(4'-(1H-Tetrazol-5-yl)-biphenyl-2-sulfonic acid (3,...)
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity to CHO cells stably expressing human Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed