Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 50011746
TargetGlucagon receptor(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50:  1nMAssay Description:Compound was evaluated in vitro for its inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110068(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110056(2,3-Dichloro-4-hydroxy-benzoic acid [1-[4-(4-isopr...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110067(2,3-Difluoro-4-hydroxy-benzoic acid [1-[4-(4-isopr...)
Affinity DataIC50:  48nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110073(4-Hydroxy-3-nitro-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110074(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  53nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110066(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-trifluoro...)
Affinity DataIC50:  58nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110055(3-Chloro-4-hydroxy-benzoic acid [1-(4-isopropyl-be...)
Affinity DataIC50:  84nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110057(3-Fluoro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110084(2-{4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110070(3-Chloro-4-hydroxy-benzoic acid [1-[4-(tetrahydro-...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110063(3-Chloro-4-hydroxy-benzoic acid [1-[4-(3,4-difluor...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110053(3-Chloro-4-hydroxy-benzoic acid [1-[4-(5-tert-buty...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110080(3-Chloro-4-hydroxy-benzoic acid [1-[3,5-dimethoxy-...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110077(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110083(3-Chloro-4-hydroxy-benzoic acid [1-[1-(4-isopropyl...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110081(CHEMBL161401 | {4-[(3-Chloro-4-hydroxy-benzoyl)-hy...)
Affinity DataIC50:  690nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110071(4-Hydroxy-benzoic acid [1-[4-(4-isopropyl-benzylox...)
Affinity DataIC50:  690nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110085(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  740nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110062(3-Chloro-4-hydroxy-benzoic acid (4-methoxy-naphtha...)
Affinity DataIC50:  870nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110060(3-Chloro-4-hydroxy-benzoic acid N'-[4-(4-isopropyl...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110076(3-Amino-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50:  940nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110065(2-{4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110082(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110078(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110069(3-Chloro-4-hydroxy-N-{2-[4-(4-isopropyl-benzyloxy)...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110058(3,4-Dihydroxy-benzoic acid [1-[4-(4-isopropyl-benz...)
Affinity DataIC50:  2.70E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110059(3-Chloro-4-hydroxy-N-{2-[4-(4-isopropyl-benzyloxy)...)
Affinity DataIC50:  5.20E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110072((E)-N-(3-Chloro-4-hydroxy-phenyl)-3-[4-(4-isopropy...)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110079(3-Cyano-4-hydroxy-benzoic acid (4-isopropyl-3,5-di...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110064(5-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl]-2...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110061(2-chloro-4-[1-[4-(4-isopropylbenzyloxy)-3,5-dimeth...)
Affinity DataIC50:  7.83E+4nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50110075(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed