Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50011962
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112639BDBM50112639(pQ-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2 | CHEMBL402688)
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112626BDBM50112626(Carbocyanine derivative | CHEMBL442514)
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112623BDBM50112623((FITC-Q-W-A-V-G-H-L-M-NH2) | CHEMBL274327)
Affinity DataIC50: 3.20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112643BDBM50112643((DTPA-P-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2) | CHEMBL442...)
Affinity DataIC50: 4.70nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112611BDBM50112611((K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL405669)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112640BDBM50112640((epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL21696...)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112629BDBM50112629((epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL38528...)
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112632BDBM50112632((alpha-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL428280)
Affinity DataIC50: 5.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112619BDBM50112619((G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL408739)
Affinity DataIC50: 7.60nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112633BDBM50112633((FITC-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL385928)
Affinity DataIC50: 9.20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112635BDBM50112635((alpha,epsilon-(-FITC)2-K-Q-W-A-V-G-H-L-M-NH2) | C...)
Affinity DataIC50: 9.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112620BDBM50112620((epsilon-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMB...)
Affinity DataIC50: 9.60nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112625BDBM50112625((K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL269310)
Affinity DataIC50: 10.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112627BDBM50112627((alpha-FITC-epsilon-DOTA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 15nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112646BDBM50112646((alpha-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL4...)
Affinity DataIC50: 15.6nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112614BDBM50112614((alpha-FITC-epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112616BDBM50112616((alpha,epsilon-(FITC)2-K-G-S-G-Q-W-A-V-G-H-L-M-NH2...)
Affinity DataIC50: 20.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112642BDBM50112642((Q-W-A-V-G-H-L-M-NH2) | CHEMBL300318)
Affinity DataIC50: 28.3nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112630BDBM50112630((alpha,epsilon-(DTPA)2-K-Q-W-A-V-G-H-L-M-NH2) | CH...)
Affinity DataIC50: 240nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112621BDBM50112621((alpha-DTPA-epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 276nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50112622BDBM50112622((alpha-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL440609)
Affinity DataIC50: 410nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed