Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 5364
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  0.930nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  1.01nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  1.11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  1.18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  1.37nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.54nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.63nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  1.65nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  1.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  2.07nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  2.49nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  2.67nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  3.92nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  4.26nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  4.81nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  4.91nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  7.87nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  8.91nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataKi:  9.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataKi:  9.57nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  10.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86029(trans-H2-PAT(+))
Affinity DataKi:  11.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataKi:  11.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM50017674(Hydramine | Benylin | Silphen | (2-Benzhydryloxy-e...)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  13.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  14.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86029(trans-H2-PAT(+))
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86029(trans-H2-PAT(+))
Affinity DataKi:  29.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86029(trans-H2-PAT(+))
Affinity DataKi:  42.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86030(cis-H2-PAT(+))
Affinity DataKi:  53.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86030(cis-H2-PAT(+))
Affinity DataKi:  77.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM81466(NSC_6445134 | CAS_23095-76-3 | l-Chlorpheniramine)
Affinity DataKi:  80.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM81466(NSC_6445134 | CAS_23095-76-3 | l-Chlorpheniramine)
Affinity DataKi:  98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86030(cis-H2-PAT(+))
Affinity DataKi:  122nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
University of North Carolina at Chapel Hill

Curated by PDSP Ki Database
LigandPNGBDBM86030(cis-H2-PAT(+))
Affinity DataKi:  129nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
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