Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50037049
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116537(3-({3-[4-(Biphenyl-4-yloxy)-phenoxy]-propyl}-methy...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116563(N-(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116562([4-(4-Benzyl-phenoxy)-butylamino]-acetic acid | CH...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116554(N-(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116560(3-{Methyl-[3-(4-thiophen-3-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116538(SC-57461A | CHEMBL543405 | CHEMBL112671 | 3-{[3-(4...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116544(2-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-eth...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116542(3-{Methyl-[3-(4-thiophen-2-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116561(3-[4-(4-Benzyl-phenoxy)-butylamino]-propionic acid...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116548(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-pro...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116532([4-(4-Benzyl-phenoxy)-butylamino]-acetic acid ethy...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116529(3-{Methyl-[3-(4-thiophen-2-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116531(3-[4-(4-Benzyl-phenoxy)-butylamino]-propionic acid...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116533(3-{Methyl-[3-(4-phenoxy-phenoxy)-propyl]-amino}-pr...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116535(3-(Methyl-{3-[4-(4-oxazol-2-yl-phenoxy)-phenoxy]-p...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116536(3-({3-[4-(4-Fluoro-benzyl)-phenoxy]-propyl}-methyl...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50085255(2-{4-[4-(2-Pyrrolidin-1-yl-ethoxy)-phenoxy]-phenyl...)
Affinity DataIC50: 43nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116538(SC-57461A | CHEMBL543405 | CHEMBL112671 | 3-{[3-(4...)
Affinity DataIC50: 49nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50085255(2-{4-[4-(2-Pyrrolidin-1-yl-ethoxy)-phenoxy]-phenyl...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116554(N-(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116553(3-(Methyl-{3-[4-(4-thiazol-2-yl-phenoxy)-phenoxy]-...)
Affinity DataIC50: 72nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116563(N-(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-...)
Affinity DataIC50: 75nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116561(3-[4-(4-Benzyl-phenoxy)-butylamino]-propionic acid...)
Affinity DataIC50: 76nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116530(3-[3-(4-Benzyl-phenoxy)-propylamino]-propionic aci...)
Affinity DataIC50: 84nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116529(3-{Methyl-[3-(4-thiophen-2-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 95nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116557({[4-(4-Benzyl-phenoxy)-butyl]-methyl-amino}-acetic...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116548(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-pro...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116559(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-pro...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116542(3-{Methyl-[3-(4-thiophen-2-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116540(3-[3-(4-Benzyl-phenoxy)-propylamino]-propionic aci...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116558(3-({3-[4-(4-Fluoro-phenoxy)-phenoxy]-propyl}-methy...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116536(3-({3-[4-(4-Fluoro-benzyl)-phenoxy]-propyl}-methyl...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116560(3-{Methyl-[3-(4-thiophen-3-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116559(3-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-pro...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116537(3-({3-[4-(Biphenyl-4-yloxy)-phenoxy]-propyl}-methy...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116535(3-(Methyl-{3-[4-(4-oxazol-2-yl-phenoxy)-phenoxy]-p...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50085251(1-[2-(Biphenyl-4-yloxy)-ethyl]-pyrrolidine | 1-[2-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116558(3-({3-[4-(4-Fluoro-phenoxy)-phenoxy]-propyl}-methy...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116546(2-{[3-(4-Benzyl-phenoxy)-propyl]-methyl-amino}-eth...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116547(3-[2-(4-Benzyl-phenoxy)-ethylamino]-propionic acid...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116562([4-(4-Benzyl-phenoxy)-butylamino]-acetic acid | CH...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116533(3-{Methyl-[3-(4-phenoxy-phenoxy)-propyl]-amino}-pr...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116545([5-(4-Benzyl-phenoxy)-pentylamino]-acetic acid eth...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116541(3-{Methyl-[3-(4-thiophen-3-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116540(3-[3-(4-Benzyl-phenoxy)-propylamino]-propionic aci...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116543(3-{Methyl-[3-(4-pyridin-3-ylmethyl-phenoxy)-propyl...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116532([4-(4-Benzyl-phenoxy)-butylamino]-acetic acid ethy...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116545([5-(4-Benzyl-phenoxy)-pentylamino]-acetic acid eth...)
Affinity DataIC50: 420nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116551(4-{[2-(4-Benzyl-phenoxy)-ethyl]-methyl-amino}-buty...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human leukotriene A4 hydrolase (LTA-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetLeukotriene A-4 hydrolase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50116557({[4-(4-Benzyl-phenoxy)-butyl]-methyl-amino}-acetic...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human whole blood LTB-4 production (Leukotriene B-4).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
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