Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50012536
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120247(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 8.5nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120236(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120246(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120257(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120237(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120269(N-[2-(4-Bromo-phenyl)-2-oxo-ethyl]-3-(2,4-dioxo-3,...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120244(N-(2-Biphenyl-4-yl-2-oxo-ethyl)-3-(2,4-dioxo-3,4,7...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120262(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120262(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120267(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120261(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120251(N-[2-(3'-Amino-biphenyl-4-yl)-2-oxo-ethyl]-3-(2,4-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120239(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120254(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120265(3-(2,4-dioxo-2,3,4,5,7,8-hexahydro-1H-thiopyrano[4...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120242(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120274(3-(2,4-Dioxo-3,4,5,6,7,8-hexahydro-2H-quinazolin-1...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120256(N-[2-(4-Difluoromethoxy-phenyl)-2-oxo-ethyl]-3-(2,...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120277(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120253(Benzoic acid 4-{2-[3-(2,4-dioxo-3,4,7,8-tetrahydro...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120238(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 30nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using dose-response inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120241(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120272(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120249(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120266(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120273(2-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120260(N-[2-(4-Chloro-phenyl)-2-oxo-ethyl]-3-(2,4-dioxo-3...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120269(N-[2-(4-Bromo-phenyl)-2-oxo-ethyl]-3-(2,4-dioxo-3,...)
Affinity DataEC50:  70nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120235(N-(2-Biphenyl-3-yl-2-oxo-ethyl)-3-(2,4-dioxo-3,4,7...)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120240(N-{2-[4-(3-Amino-pyridin-2-yl)-piperazin-1-yl]-2-o...)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120262(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  70nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120262(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  70nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120254(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  70nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120252(N-[2-(3-Bromo-phenyl)-2-oxo-ethyl]-3-(2,4-dioxo-3,...)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120251(N-[2-(3'-Amino-biphenyl-4-yl)-2-oxo-ethyl]-3-(2,4-...)
Affinity DataEC50:  70nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120265(3-(2,4-dioxo-2,3,4,5,7,8-hexahydro-1H-thiopyrano[4...)
Affinity DataEC50:  80nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120268(N-[2-(4-Bromo-phenyl)-2-oxo-ethyl]-3-(2,4-dioxo-3,...)
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120247(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  80nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120278(3-(2,4-Dioxo-3,4,5,6,7,8-hexahydro-2H-quinazolin-1...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120237(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120238(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120246(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120267(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120241(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120239(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant Poly (ADP-ribose) polymerase 1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120272(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  100nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120255(2-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120243(3-(2,4-Dioxo-3,4,5,6,7,8-hexahydro-2H-quinazolin-1...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against human recombinant PARP-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120256(N-[2-(4-Difluoromethoxy-phenyl)-2-oxo-ethyl]-3-(2,...)
Affinity DataEC50:  200nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50120236(3-(2,4-Dioxo-3,4,7,8-tetrahydro-2H,5H-thiopyrano[4...)
Affinity DataEC50:  200nMAssay Description:Concentration required to inhibit human recombinant PARP-1 was determined using cell protection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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