Compile Data Set for Download or QSAR
Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 50012709
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121759BDBM50121759([D-Leu15]orexin-B | CHEMBL438587)
Affinity DataEC50:  0.0520nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121770BDBM50121770([Ala14]orexin-B | CHEMBL413504)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121788BDBM50121788([Ala11]orexin-B | CHEMBL441918)
Affinity DataEC50:  0.0660nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121783BDBM50121783(Orexin-B | CHEMBL413434)
Affinity DataEC50:  0.0810nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121775BDBM50121775([D-Leu7]orexin-B | CHEMBL438036)
Affinity DataEC50:  0.0840nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121795BDBM50121795([Gly17]orexin-B | CHEMBL436915)
Affinity DataEC50:  0.0910nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121769BDBM50121769([D-Gln12]orexin-B | CHEMBL428123)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121815BDBM50121815([Ala6]orexin-B | CHEMBL410480)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121794BDBM50121794([Ala7]orexin-B | CHEMBL427771)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121796BDBM50121796([Ala16]orexin-B | CHEMBL414312)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121810BDBM50121810([D-Ala9]orexin-B | CHEMBL409301)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121765BDBM50121765([Ala13]orexin-B | CHEMBL437464)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121791BDBM50121791([D-Pro4]orexin-B | CHEMBL410947)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121777BDBM50121777([D-Ser2]orexin-B | CHEMBL265746)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121817BDBM50121817([Trp11]orexin-B | CHEMBL437149)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121778BDBM50121778([D-Ala3]orexin-B | CHEMBL265423)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121792BDBM50121792([D-Ala19]orexin-B | CHEMBL439541)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121809BDBM50121809([D-Pro5]orexin-B | CHEMBL410899)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121803BDBM50121803([Ala3]orexin-B | CHEMBL265404)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121766BDBM50121766([D-Arg1]orexin-B | CHEMBL410816)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121793BDBM50121793([D-Ala6]orexin-B | CHEMBL264342)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121790BDBM50121790([Ala1]orexin-B | CHEMBL409456)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121806BDBM50121806([Ala9]orexin-B | CHEMBL265907)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121780BDBM50121780([Ala2]orexin-B | CHEMBL414332)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121784BDBM50121784([Ala12]orexin-B | CHEMBL266409)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121797BDBM50121797([Ala4]orexin-B | CHEMBL437274)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121773BDBM50121773([D-Asn20]orexin-B | CHEMBL386549)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121767BDBM50121767([D-Ala17]orexin-B | CHEMBL409970)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121781BDBM50121781([Gly22]orexin-B | CHEMBL275985)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121786BDBM50121786([Ala5]orexin-B | CHEMBL442505)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121772BDBM50121772([D-Gln8]orexin-B | CHEMBL413284)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121795BDBM50121795([Gly17]orexin-B | CHEMBL436915)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121760BDBM50121760([D-Gln16]orexin-B | CHEMBL413285)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121785BDBM50121785([D-Arg13]orexin-B | CHEMBL411174)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121800BDBM50121800([D-Leu14]orexin-B | CHEMBL409697)
Affinity DataEC50:  0.440nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121764BDBM50121764([D-Ser18]orexin-B | CHEMBL411116)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121761BDBM50121761([Ala8]orexin-B | CHEMBL441008)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121792BDBM50121792([D-Ala19]orexin-B | CHEMBL439541)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121774BDBM50121774([D-Leu11]orexin-B | CHEMBL264343)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121773BDBM50121773([D-Asn20]orexin-B | CHEMBL386549)
Affinity DataEC50:  0.610nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121798BDBM50121798([Ala21]orexin-B | CHEMBL413884)
Affinity DataEC50:  0.720nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121805BDBM50121805([Ala10]orexin-B | CHEMBL430064)
Affinity DataEC50:  0.770nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121769BDBM50121769([D-Gln12]orexin-B | CHEMBL428123)
Affinity DataEC50:  0.770nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121770BDBM50121770([Ala14]orexin-B | CHEMBL413504)
Affinity DataEC50:  0.820nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121783BDBM50121783(Orexin-B | CHEMBL413434)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121799BDBM50121799([Gly23]orexin-B | CHEMBL409967)
Affinity DataEC50:  0.840nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121809BDBM50121809([D-Pro5]orexin-B | CHEMBL410899)
Affinity DataEC50:  0.850nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121763BDBM50121763([D-Arg10]orexin-B | CHEMBL410960)
Affinity DataEC50:  0.870nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121791BDBM50121791([D-Pro4]orexin-B | CHEMBL410947)
Affinity DataEC50:  0.890nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121776BDBM50121776([D-His21]orexin-B | CHEMBL430313)
Affinity DataEC50:  1nMAssay Description:Agonist activity against human orexin 2 receptor; EC50; nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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