Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50048560
LigandPNGBDBM50222081(CHEMBL327654)
Affinity DataKi:  5.10nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  6.20nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  10nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  11nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50130287((4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222053(CHEMBL90752)
Affinity DataKi:  18nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50130287((4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-...)
Affinity DataKi:  19nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222053(CHEMBL90752)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222082(CHEMBL544315)
Affinity DataKi:  22nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  24nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222083(CHEMBL90538)
Affinity DataKi:  26nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222047(CHEMBL316283)
Affinity DataKi:  26nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  26nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222047(CHEMBL316283)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222083(CHEMBL90538)
Affinity DataKi:  28nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222048(CHEMBL540821)
Affinity DataKi:  32nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222050(CHEMBL92856)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222056(CHEMBL94017)
Affinity DataKi:  44nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222049(CHEMBL90150)
Affinity DataKi:  46nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222051(CHEMBL90118)
Affinity DataKi:  69nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222050(CHEMBL92856)
Affinity DataKi:  74nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222049(CHEMBL90150)
Affinity DataKi:  79nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222048(CHEMBL540821)
Affinity DataKi:  89nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222082(CHEMBL544315)
Affinity DataKi:  91nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222052(CHEMBL329548)
Affinity DataKi:  102nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50222054(CHEMBL94056)
Affinity DataKi:  110nMAssay Description:Affinity for Alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222055(CHEMBL327906)
Affinity DataKi:  132nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222048(CHEMBL540821)
Affinity DataKi:  155nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222053(CHEMBL90752)
Affinity DataKi:  166nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222082(CHEMBL544315)
Affinity DataKi:  170nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222054(CHEMBL94056)
Affinity DataKi:  182nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50130287((4,5-Dihydro-1H-imidazol-2-yl)-(2-methyl-biphenyl-...)
Affinity DataKi:  209nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222050(CHEMBL92856)
Affinity DataKi:  209nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222081(CHEMBL327654)
Affinity DataKi:  257nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222081(CHEMBL327654)
Affinity DataKi:  257nMAssay Description:Inhibition of [3H]-5-CT binding to 5-hydroxytryptamine 7 receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222049(CHEMBL90150)
Affinity DataKi:  257nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222047(CHEMBL316283)
Affinity DataKi:  263nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222083(CHEMBL90538)
Affinity DataKi:  275nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50222054(CHEMBL94056)
Affinity DataKi:  1.20E+3nMAssay Description:Affinity for Alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed