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Found 12 Enz. Inhib. hit(s) with all data for entry = 50042007
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  2.21E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50005628((S) Verapamil | (S)-5-((3,4-dimethoxyphenethyl)(me...)
Affinity DataIC50:  2.44E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50338982((R)-5-((3,4-dimethoxyphenethyl)(methyl)amino)-2-(3...)
Affinity DataIC50:  2.58E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420194(CHEMBL2074950)
Affinity DataIC50:  3.04E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420195(CHEMBL2074951)
Affinity DataIC50:  3.11E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420194(CHEMBL2074950)
Affinity DataIC50:  3.20E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in HCT15/CL02 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  4.78E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50005628((S) Verapamil | (S)-5-((3,4-dimethoxyphenethyl)(me...)
Affinity DataIC50:  5.33E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50338982((R)-5-((3,4-dimethoxyphenethyl)(methyl)amino)-2-(3...)
Affinity DataIC50:  5.52E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420194(CHEMBL2074950)
Affinity DataIC50:  6.63E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420194(CHEMBL2074950)
Affinity DataIC50:  7.63E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50420195(CHEMBL2074951)
Affinity DataIC50:  7.65E+3nMAssay Description:TP_TRANSPORTER: drug resistance (paclitaxel) in MES-SA/DX5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed