Compile Data Set for Download or QSAR
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Found 43 Enz. Inhib. hit(s) with all data for entry = 50012902
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124076((S)-1-((R)-3-Cyclohexyl-1-oxo-2-phenylmethanesulfo...)
Affinity DataKi:  140nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124071(((R)-1-Cyclohexylmethyl-2-oxo-2-{(S)-2-[(4,5,6,7-t...)
Affinity DataKi:  280nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124073((S)-1-((R)-2-Amino-1-oxo-3,3-diphenyl-propyl)-pyrr...)
Affinity DataKi:  360nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124083(((R)-1-Benzhydryl-2-oxo-2-{(S)-2-[(4,5,6,7-tetrahy...)
Affinity DataKi:  530nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124075((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-1-oxo-p...)
Affinity DataKi:  690nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124077(((R)-1-(3,4-Dichloro-benzyl)-2-oxo-2-{(S)-2-[(4,5,...)
Affinity DataKi:  3.33E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124072(((R)-2-{(S)-2-[(2-Amino-5,6,7,8-tetrahydro-quinazo...)
Affinity DataKi:  4.50E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124078((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  5.38E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124074((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  1.28E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124084((S)-1-((R)-2-Amino-3,3-diphenyl-propionyl)-pyrroli...)
Affinity DataKi:  1.29E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124071(((R)-1-Cyclohexylmethyl-2-oxo-2-{(S)-2-[(4,5,6,7-t...)
Affinity DataKi:  1.99E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124085((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  2.73E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124082((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >3.51E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124079((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >3.51E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124081(CHEMBL164221 | [(R)-2-{(S)-2-[(2-Amino-5,6,7,8-tet...)
Affinity DataKi: >3.51E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124080((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-propion...)
Affinity DataKi: >3.51E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124084((S)-1-((R)-2-Amino-3,3-diphenyl-propionyl)-pyrroli...)
Affinity DataKi:  5.76E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124079((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124078((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124075((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-1-oxo-p...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124082((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124080((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-propion...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124076((S)-1-((R)-3-Cyclohexyl-1-oxo-2-phenylmethanesulfo...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124077(((R)-1-(3,4-Dichloro-benzyl)-2-oxo-2-{(S)-2-[(4,5,...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124081(CHEMBL164221 | [(R)-2-{(S)-2-[(2-Amino-5,6,7,8-tet...)
Affinity DataKi: >6.83E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124076((S)-1-((R)-3-Cyclohexyl-1-oxo-2-phenylmethanesulfo...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124080((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-propion...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124078((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124079((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124082((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124077(((R)-1-(3,4-Dichloro-benzyl)-2-oxo-2-{(S)-2-[(4,5,...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124075((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-1-oxo-p...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124081(CHEMBL164221 | [(R)-2-{(S)-2-[(2-Amino-5,6,7,8-tet...)
Affinity DataKi: >7.54E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124073((S)-1-((R)-2-Amino-1-oxo-3,3-diphenyl-propyl)-pyrr...)
Affinity DataKi:  8.21E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124071(((R)-1-Cyclohexylmethyl-2-oxo-2-{(S)-2-[(4,5,6,7-t...)
Affinity DataKi:  8.48E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124083(((R)-1-Benzhydryl-2-oxo-2-{(S)-2-[(4,5,6,7-tetrahy...)
Affinity DataKi:  8.52E+4nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124070((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  1.11E+5nMAssay Description:In vitro inhibitory activity of the compound against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124073((S)-1-((R)-2-Amino-1-oxo-3,3-diphenyl-propyl)-pyrr...)
Affinity DataKi:  2.17E+5nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124070((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  2.89E+5nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124070((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  3.42E+5nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124084((S)-1-((R)-2-Amino-3,3-diphenyl-propionyl)-pyrroli...)
Affinity DataKi:  4.09E+5nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124085((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  4.16E+5nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124074((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  7.30E+5nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed