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Found 9 Enz. Inhib. hit(s) with all data for entry = 50013105
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(CHEMBL263595 | Compound [Gly2]Venorphin)
Affinity DataKi:  8.40nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 using [3H]-Diprenorphine as radioligand in Chinese hamster ovary cells expressing cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(CHEMBL438571 | Compound Venorphin)
Affinity DataKi:  20nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 using [3H]-Diprenorphine as radioligand in Chinese hamster ovary cells expressing cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(CHEMBL414369 | cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-A...)
Affinity DataKi:  27nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 using [3H]-Diprenorphine as radioligand in Chinese hamster ovary cells expressing cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(CHEMBL438571 | Compound Venorphin)
Affinity DataKi:  251nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 using [3H]-DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(CHEMBL414369 | cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-A...)
Affinity DataKi:  331nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 using [3H]-DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(CHEMBL263595 | Compound [Gly2]Venorphin)
Affinity DataKi:  339nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 using [3H]-DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(CHEMBL438571 | Compound Venorphin)
Affinity DataKi:  5.32E+3nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 using [3H]-DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(CHEMBL414369 | cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-A...)
Affinity DataKi: >8.90E+3nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 using [3H]-DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(CHEMBL263595 | Compound [Gly2]Venorphin)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 using [3H]-DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed