Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50003642
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataKi:  34nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50170163(CHEMBL321860)
Affinity DataKi:  126nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474242(CHEMBL106931)
Affinity DataKi:  219nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474249(CHEMBL106158)
Affinity DataKi:  224nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474240(Imifuramine)
Affinity DataKi:  229nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474250(CHEMBL105803)
Affinity DataKi:  245nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474252(CHEMBL320331)
Affinity DataKi:  331nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474252(CHEMBL320331)
Affinity DataKi:  437nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474240(Imifuramine)
Affinity DataKi:  891nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474247(CHEMBL109130)
Affinity DataKi:  1.02E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474250(CHEMBL105803)
Affinity DataKi:  1.05E+3nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474244(CHEMBL106913)
Affinity DataKi:  1.70E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474248(CHEMBL321920)
Affinity DataKi:  2.04E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50170163(CHEMBL321860)
Affinity DataKi:  2.19E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474248(CHEMBL321920)
Affinity DataKi:  2.51E+3nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi:  2.51E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474244(CHEMBL106913)
Affinity DataKi:  6.46E+3nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474253(CHEMBL1632410)
Affinity DataKi:  6.92E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474249(CHEMBL106158)
Affinity DataKi:  7.08E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474251(CHEMBL108649)
Affinity DataKi:  8.13E+3nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474251(CHEMBL108649)
Affinity DataKi:  8.13E+3nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474241(CHEMBL322256)
Affinity DataKi:  1.05E+4nMAssay Description:Compound was tested for H3 receptor competition binding using [3H]- Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474245(CHEMBL320279)
Affinity DataKi:  1.15E+4nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474247(CHEMBL109130)
Affinity DataKi:  1.17E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataKi:  1.20E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474242(CHEMBL106931)
Affinity DataKi:  1.29E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474253(CHEMBL1632410)
Affinity DataKi:  1.35E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474243(CHEMBL106570)
Affinity DataKi:  1.86E+4nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474239(CHEMBL107877)
Affinity DataKi:  2.00E+4nMAssay Description:Compound was tested for H3 receptor competition binding using [3H]- Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474243(CHEMBL106570)
Affinity DataKi:  2.04E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474241(CHEMBL322256)
Affinity DataKi:  2.14E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474245(CHEMBL320279)
Affinity DataKi:  2.19E+4nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataKi: <1.00E+5nMAssay Description:Histamine H4 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474243(CHEMBL106570)
Affinity DataEC50: <1.00E+5nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474244(CHEMBL106913)
Affinity DataEC50:  813nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474245(CHEMBL320279)
Affinity DataEC50:  4.07E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474241(CHEMBL322256)
Affinity DataEC50:  1.29E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474247(CHEMBL109130)
Affinity DataEC50:  269nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474244(CHEMBL106913)
Affinity DataEC50:  7.59E+3nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM81542(Beta-Methylhistamine | CAS_565544 | NSC_565544)
Affinity DataEC50:  0.123nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataEC50:  21nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50170163(CHEMBL321860)
Affinity DataEC50:  78nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474249(CHEMBL106158)
Affinity DataEC50:  224nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474248(CHEMBL321920)
Affinity DataEC50:  5.50E+3nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474250(CHEMBL105803)
Affinity DataEC50:  91nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474252(CHEMBL320331)
Affinity DataEC50:  191nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474246(CHEMBL319658)
Affinity DataEC50:  8.51E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474249(CHEMBL106158)
Affinity DataEC50:  1.02E+4nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474242(CHEMBL106931)
Affinity DataEC50:  105nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50474250(CHEMBL105803)
Affinity DataEC50:  741nMAssay Description:Inhibition of the forskolin-stimulated cAMP production in SK-N-MC cells expressing human Histamine H4 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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