Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50013441
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130611(2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130617(2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130619(2-Amino-N-{8-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130613(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130612(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130614(2-Amino-N-{2-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130619(2-Amino-N-{8-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  15nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130617(2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  46nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130611(2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  53nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130612(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataKi:  62nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130614(2-Amino-N-{2-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataKi:  116nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130613(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  133nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130618(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  309nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130615(2-Amino-N-{8-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  399nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130621(2-Amino-N-{6-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  410nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130620(2-Amino-N-{2-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  648nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130616(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataKi:  1.53E+3nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130615(2-Amino-N-{8-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  6.15E+3nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130618(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  6.50E+3nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130620(2-Amino-N-{2-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  8.29E+3nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130621(2-Amino-N-{6-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataKi:  2.19E+4nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130616(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataKi:  4.62E+4nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130617(2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50:  3.10nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130611(2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50:  5.30nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130619(2-Amino-N-{8-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50:  54nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130612(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataIC50:  181nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130613(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataIC50:  255nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130614(2-Amino-N-{2-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50:  2.84E+3nMAssay Description:Opioid receptor mu 1 agonism in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130613(2-Amino-N-{4-[2-amino-3-(4-hydroxy-phenyl)-propion...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130611(2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130619(2-Amino-N-{8-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130617(2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130612(2-Amino-N-[4-(2-amino-3-phenyl-propionylamino)-but...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50130614(2-Amino-N-{2-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Opioid receptor delta 1 agonism in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed