Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50013482
LigandPNGBDBM50131110(CHEMBL437226 | Cyclic peptide analogue)
Affinity DataIC50:  420nMAssay Description:Inhibition of Farnesyltransferase by Scintillation Proximity AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50131111(CHEMBL87258 | H-SMGLPCVVM-OH)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Farnesyltransferase by Scintillation Proximity AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50131111(CHEMBL87258 | H-SMGLPCVVM-OH)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of farnesylation of v-Ki-Ras by bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50131112(CHEMBL410280 | Cyclic peptide analogue)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibition of mouse melanoma B16-F10 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50131110(CHEMBL437226 | Cyclic peptide analogue)
Affinity DataIC50:  5.60E+5nMAssay Description:Inhibition of mouse melanoma B16-F10 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50131113(CHEMBL410479 | Cyclic peptide analogue)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibition of mouse melanoma B16-F10 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50131108(CHEMBL402695 | H-VYAVTGRGDSPA-NH2)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of mouse melanoma B16-F10 cell adhesion to fibronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50131109((S)-3-[2-((S)-2-{2-[(2S,3R)-2-((S)-2-Amino-3-methy...)
Affinity DataIC50:  1.10E+6nMAssay Description:In vitro inhibition of farnesylation of v-Ki-Ras by bovine farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed