Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50048882
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229974(CHEMBL178077)
Affinity DataIC50:  452nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  603nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229967(CHEMBL263944)
Affinity DataIC50:  666nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229969(CHEMBL554645)
Affinity DataIC50:  727nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229970(CHEMBL367876)
Affinity DataIC50:  796nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229972(CHEMBL174721)
Affinity DataIC50:  929nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229966(DESMETHYL-OFLOXACIN | Desmethyl-Ofloxacin (5%))
Affinity DataIC50:  1.69E+3nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50229965(CHEMBL174892)
Affinity DataIC50:  2.58E+3nMAssay Description:The inhibitory activity was measured for the supercoiling activity of DNA gyrase isolated from Escherichia coli K-12 C600.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed