Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50000025
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000438(CHEMBL355389 | 5-(4-Dimethylamino-phenylcarbamoyl)...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000430(CHEMBL167145 | 5-(4-Ethoxy-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM26114(CHEMBL88972 | pyridine-2,5-dicarboxylic acid | pyr...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000437(CHEMBL424388 | 5-p-Tolylcarbamoyl-pyridine-2-carbo...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000417(CHEMBL167904 | 5-(2-Fluoro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000429(CHEMBL353753 | 5-(4-Ethoxy-benzoylamino)-pyridine-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000420(CHEMBL165333 | 5-(4-Dimethylamino-benzoylamino)-py...)
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000433(CHEMBL165533 | 5-(2-Methoxy-phenylcarbamoyl)-pyrid...)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000424(CHEMBL354140 | 5-(4-Fluoro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000441(CHEMBL352785 | 5-(2-Chloro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000434(CHEMBL167789 | 5-(4-Methyl-benzoylamino)-pyridine-...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000436(CHEMBL353379 | 5-(2,4-Dimethoxy-phenylcarbamoyl)-p...)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000432(CHEMBL166382 | 5-(4-Chloro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 1.74E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000442(CHEMBL167209 | 5-(4-Methoxy-phenylcarbamoyl)-pyrid...)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000435(CHEMBL167699 | 5-(4-Chloro-benzoylamino)-pyridine-...)
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000428(CHEMBL30897 | 5-Benzoylamino-pyridine-2-carboxylic...)
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000421(CHEMBL167574 | 5-(3,4,5-Trimethoxy-phenylcarbamoyl...)
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000440(CHEMBL354059 | 5-Phenylcarbamoyl-pyridine-2-carbox...)
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000423(CHEMBL30729 | 5-(4-Fluoro-benzylamino)-pyridine-2-...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000419(CHEMBL167097 | 5-(3-Chloro-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000418(CHEMBL167756 | 5-(2-Ethoxy-phenylcarbamoyl)-pyridi...)
Affinity DataIC50: 3.29E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000427(CHEMBL167725 | 5-(2-Fluoro-benzoylamino)-pyridine-...)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000431(CHEMBL166172 | 5-Benzyloxy-pyridine-2-carboxylic a...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000422(CHEMBL166105 | 5-(4-Nitro-phenylcarbamoyl)-pyridin...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000426(CHEMBL167946 | 5-(4-Fluoro-benzoylamino)-pyridine-...)
Affinity DataIC50: 5.12E+4nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000423(CHEMBL30729 | 5-(4-Fluoro-benzylamino)-pyridine-2-...)
Affinity DataIC50: 8.00E+4nMAssay Description:Compound was evaluated for inhibition of Prolyl 4-hydroxylase activity in cultured embryonic chick tendon cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000439(CHEMBL24510 | 5-Butyl-pyridine-2-carboxylic acid |...)
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransmembrane prolyl 4-hydroxylase(Human)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000425(CHEMBL167489 | 5-[2-(4-Chloro-phenyl)-vinyl]-pyrid...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of prolyl 4-hydroxylase activity by an indirect assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed