Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50000055
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000714BDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataKi:  98nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000717BDBM50000717(CHEMBL65132 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  142nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000701BDBM50000701(CHEMBL264497 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-...)
Affinity DataKi:  157nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000707BDBM50000707(CHEMBL62873 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  167nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000722BDBM50000722(CHEMBL63111 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  331nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000720BDBM50000720(CHEMBL66414 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  345nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000719BDBM50000719(CHEMBL62812 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...)
Affinity DataKi:  390nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000708BDBM50000708(CHEMBL64094 | 4-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  656nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000700BDBM50000700(CHEMBL66537 | 4-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  690nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000716BDBM50000716(CHEMBL61680 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...)
Affinity DataKi:  925nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000718BDBM50000718(CHEMBL65144 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  945nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000705BDBM50000705(CHEMBL65228 | 2-({7-[4-(4-Fluoro-phenyl)-1-methyl-...)
Affinity DataKi:  1.58E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000712BDBM50000712(CHEMBL303312 | 7-[4-(4-Fluoro-phenyl)-1-methyl-but...)
Affinity DataKi:  3.25E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000711BDBM50000711(CHEMBL61014 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  3.30E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000715BDBM50000715(CHEMBL304427 | 2-[7-(1,2-Dimethyl-heptyl)-5-hydrox...)
Affinity DataKi:  3.68E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000702BDBM50000702(CHEMBL65556 | 7-[4-(4-Fluoro-phenyl)-1-methyl-buty...)
Affinity DataKi:  4.21E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000710BDBM50000710(CHEMBL62650 | 3-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  4.40E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000709BDBM50000709(CHEMBL65199 | 5-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000699BDBM50000699(CHEMBL61678 | 3-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000724BDBM50000724(CHEMBL65089 | 2-(5-Hydroxy-7-isopropyl-10,10-dimet...)
Affinity DataKi:  9.00E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000725BDBM50000725(CHEMBL62822 | 7-[4-(4-Fluoro-phenyl)-1-methyl-buty...)
Affinity DataKi:  1.18E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000721BDBM50000721(CHEMBL302863 | 2-{7-[4-(4-Fluoro-phenyl)-1-methyl-...)
Affinity DataKi:  1.58E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000703BDBM50000703(CHEMBL62322 | 7-[4-(4-Fluoro-phenyl)-1-methyl-buty...)
Affinity DataKi:  1.69E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000723BDBM50000723(CHEMBL62503 | 1-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  2.05E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000726BDBM50000726(CHEMBL65377 | 4-{7-[4-(4-Fluoro-phenyl)-1-methyl-b...)
Affinity DataKi:  2.07E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000713BDBM50000713(CHEMBL65715 | 2-[5-{4-[4-(4-Fluoro-phenyl)-1-methy...)
Affinity DataKi:  2.35E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000706BDBM50000706(CHEMBL291432 | 6-{7-[4-(4-Fluoro-phenyl)-1-methyl-...)
Affinity DataKi:  2.50E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000704BDBM50000704(CHEMBL61627 | 7-[4-(4-Fluoro-phenyl)-1-methyl-buty...)
Affinity DataKi:  4.38E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed