Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50036105
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001974(CHEMBL11577 | 6-Dipropylamino-1,2,6,7-tetrahydro-5...)
Affinity DataKi:  2.40nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001969(CHEMBL273867 | 6-Dipropylamino-1,2,6,7-tetrahydro-...)
Affinity DataKi:  3.20nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  6.60nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368591(CHEMBL1794795)
Affinity DataKi:  12nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368582(CHEMBL1794997)
Affinity DataKi:  13nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001977(CHEMBL269419 | 6-Dipropylamino-6,7-dihydro-5H-pyri...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368584(CHEMBL1202415)
Affinity DataKi:  30nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368593(CHEMBL1202416)
Affinity DataKi:  31nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368594(CHEMBL1794998)
Affinity DataKi:  35nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001979(CHEMBL12157 | 5-Dipropylamino-5,6-dihydro-1H,4H-im...)
Affinity DataKi:  40nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368590(CHEMBL1202409)
Affinity DataKi:  44nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKi:  46nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001971(CHEMBL268274 | 6-Dipropylamino-1,2,6,7-tetrahydro-...)
Affinity DataKi:  49nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataKi:  54nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from Dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368595(CHEMBL1744080)
Affinity DataKi:  68nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from Dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001971(CHEMBL268274 | 6-Dipropylamino-1,2,6,7-tetrahydro-...)
Affinity DataKi:  80nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001974(CHEMBL11577 | 6-Dipropylamino-1,2,6,7-tetrahydro-5...)
Affinity DataKi:  83nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368592(CHEMBL1202412)
Affinity DataKi:  84nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001979(CHEMBL12157 | 5-Dipropylamino-5,6-dihydro-1H,4H-im...)
Affinity DataKi:  90nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368595(CHEMBL1744080)
Affinity DataKi:  92nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368588(CHEMBL1202413)
Affinity DataKi:  94nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001964(CHEMBL273711 | 5-(Bis-cyclopropylmethyl-amino)-5,6...)
Affinity DataKi:  95nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368587(CHEMBL1202407)
Affinity DataKi:  102nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368594(CHEMBL1794998)
Affinity DataKi:  105nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001976(CHEMBL11896 | 5-Dipropylamino-5,6-dihydro-1H,4H-py...)
Affinity DataKi:  108nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368586(CHEMBL1202410)
Affinity DataKi:  109nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001972(CHEMBL12515 | 5-Dipropylamino-1-methyl-5,6-dihydro...)
Affinity DataKi:  124nMAssay Description:Compound was evaluated for its ability to displace [3H]DPAT from 5-HT1A receptor in homogenates of bovine hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368596(CHEMBL1202414)
Affinity DataKi:  150nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001978(CHEMBL12021 | 5-(Butyl-propyl-amino)-5,6-dihydro-1...)
Affinity DataKi:  167nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001978(CHEMBL12021 | 5-(Butyl-propyl-amino)-5,6-dihydro-1...)
Affinity DataKi:  171nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001958(CHEMBL267107 | (2-Methylsulfanyl-5,6-dihydro-4H-im...)
Affinity DataKi:  173nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368587(CHEMBL1202407)
Affinity DataKi:  207nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368583(CHEMBL1794999)
Affinity DataKi:  210nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368583(CHEMBL1794999)
Affinity DataKi:  252nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368593(CHEMBL1202416)
Affinity DataKi:  292nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368584(CHEMBL1202415)
Affinity DataKi:  304nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001977(CHEMBL269419 | 6-Dipropylamino-6,7-dihydro-5H-pyri...)
Affinity DataKi:  315nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368589(CHEMBL1202411)
Affinity DataKi:  350nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368586(CHEMBL1202410)
Affinity DataKi:  363nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKi:  534nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50453287(CHEMBL2092845)
Affinity DataKi:  569nMAssay Description:Compound was evaluated for its ability to displace [3H]DPAT from 5-HT1A receptor in homogenates of bovine hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001966(CHEMBL274419 | 5-Dipropylamino-5,6-dihydro-4H-pyrr...)
Affinity DataKi:  687nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001962(CHEMBL417612 | (5,6-Dihydro-4H-imidazo[4,5,1-ij]qu...)
Affinity DataKi:  827nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001957(CHEMBL11729 | 5-Dipropylamino-5,6-dihydro-4H-oxazo...)
Affinity DataKi:  899nMAssay Description:Ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001972(CHEMBL12515 | 5-Dipropylamino-1-methyl-5,6-dihydro...)
Affinity DataKi:  924nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from Dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001980(CHEMBL275572 | 6-Dipropylamino-6,7-dihydro-5H-pyri...)
Affinity DataKi:  933nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368585(CHEMBL1202408)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from Dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50453287(CHEMBL2092845)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from Dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50001987(CHEMBL441331 | 5-Diallylamino-5,6-dihydro-1H,4H-im...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50368596(CHEMBL1202414)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-DPAT from 5-hydroxytryptamine 1A receptor in homogenates of bovine hippocampus.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
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