Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50013871
Target72 kDa type IV collagenase(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.104nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.191nMAssay Description:Inhibition of human matrix metalloprotease-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135601(N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135602(N*1*-{2-[2-(2-Dimethylamino-ethyl)-1H-indol-3-yl]-...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135600((S)-2-((E)-2-Hydroxycarbamoylmethyl-4-methyl-pent-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50451552(CHEMBL2111573)
Affinity DataIC50: 20nMAssay Description:Inhibition of human matrix metalloprotease-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135601(N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 179nMAssay Description:Inhibition of human matrix metalloprotease-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135602(N*1*-{2-[2-(2-Dimethylamino-ethyl)-1H-indol-3-yl]-...)
Affinity DataIC50: 665nMAssay Description:Inhibition of human matrix metalloprotease-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50451552(CHEMBL2111573)
Affinity DataIC50: 910nMAssay Description:Inhibition of human matrix metalloprotease-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Umr/Cnrs 6013

Curated by ChEMBL
LigandPNGBDBM50135600((S)-2-((E)-2-Hydroxycarbamoylmethyl-4-methyl-pent-...)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of human matrix metalloprotease-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed