Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50037215
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataKi:  400nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataKi:  5.25E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135847(Bicyclic Guanidinium Subunit | CHEMBL404936)
Affinity DataKi:  7.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135843(Bicyclic Guanidinium Subunit | CHEMBL216653)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135843(Bicyclic Guanidinium Subunit | CHEMBL216653)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135846(Bicyclic Guanidinium Subunit | CHEMBL428283)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135847(Bicyclic Guanidinium Subunit | CHEMBL404936)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50135848(Bicyclic Guanidinium Subunit | CHEMBL414980)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro inhibitory activity against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed