Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 1187
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9797BDBM9797(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  0.590nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9782BDBM9782((2S)-6-{2-[benzyl(phenyl)amino]acetamido}-2-[(4-me...)
Affinity DataKi:  0.720nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9804BDBM9804(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  1.10nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9799BDBM9799(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  1.20nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9798BDBM9798(N-[(5S)-6-hydroxy-5-[(4-methylbenzene)(2-methylpro...)
Affinity DataKi:  1.40nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9784BDBM9784((2S)-6-[(2S)-2-amino-3-phenylpropanamido]-2-[(4-me...)
Affinity DataKi:  1.5nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9801BDBM9801(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  1.5nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9794BDBM9794(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  1.60nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9785BDBM9785((2S)-6-[(2S)-2-(methylamino)-3-phenylpropanamido]-...)
Affinity DataKi:  2.10nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9802BDBM9802(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  2.30nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9803BDBM9803(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  2.30nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9792BDBM9792(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  2.40nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9793BDBM9793(2-{[(2,3-dimethoxyphenyl)methyl](phenyl)amino}-N-[...)
Affinity DataKi:  2.40nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9787BDBM9787(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  2.40nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9796BDBM9796(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  2.90nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9795BDBM9795(2-{[(3,4-dimethoxyphenyl)methyl](phenyl)amino}-N-[...)
Affinity DataKi:  3.5nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9800BDBM9800(N-[(5S)-6-hydroxy-5-[(4-methylbenzene)(2-methylpro...)
Affinity DataKi:  3.90nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9774BDBM9774((2S)-6-[(2S)-2-hydroxy-3-phenylpropanamido]-2-[(4-...)
Affinity DataKi:  6.20nM ΔG°:  -47.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9806BDBM9806(N-[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfona...)
Affinity DataKi:  6.90nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9766BDBM9766((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi:  6.90nM ΔG°:  -47.4kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9791BDBM9791(N-[(5S)-6-hydroxy-5-[(4-methylbenzene)(2-methylpro...)
Affinity DataKi:  7.30nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9786BDBM9786(2-[benzyl(phenyl)amino]-N-[(5S)-6-hydroxy-5-[(4-me...)
Affinity DataKi:  7.60nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9805BDBM9805(2-{[(3-aminophenyl)methyl](phenyl)amino}-N-[(5S)-6...)
Affinity DataKi:  7.60nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9778BDBM9778((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi:  7.80nM ΔG°:  -47.1kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9783BDBM9783((2S)-6-[(dibenzylcarbamoyl)amino]-2-[(4-methylbenz...)
Affinity DataKi:  8nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9790BDBM9790(2-(diphenylamino)-N-[(5S)-6-hydroxy-5-[(4-methylbe...)
Affinity DataKi:  12nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9780BDBM9780((2S)-6-{2-[methyl(phenyl)amino]acetamido}-2-[(4-me...)
Affinity DataKi:  12nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9775BDBM9775((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi:  14nM ΔG°:  -45.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9789BDBM9789(N-[(5S)-6-hydroxy-5-[(4-methylbenzene)(2-methylpro...)
Affinity DataKi:  16nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9776BDBM9776((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi:  18nM ΔG°:  -44.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9773BDBM9773((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi:  18nM ΔG°:  -44.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9777BDBM9777((2S)-6-[2-(benzenesulfonyl)acetamido]-2-[(4-methyl...)
Affinity DataKi:  20nM ΔG°:  -44.7kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9779BDBM9779((2S)-6-[(benzylcarbamoyl)amino]-2-[(4-methylbenzen...)
Affinity DataKi:  32nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9788BDBM9788(N-[(5S)-6-hydroxy-5-[(4-methylbenzene)(2-methylpro...)
Affinity DataKi:  52nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9781BDBM9781((2S)-6-{[benzyl(methyl)carbamoyl]amino}-2-[(4-meth...)
Affinity DataKi:  55nMAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9770BDBM9770((2S)-6-(1,1-diphenylacetamido)-2-[(4-methylbenzene...)
Affinity DataKi:  171nM ΔG°:  -39.3kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9764BDBM9764((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9765BDBM9765((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9767BDBM9767((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9768BDBM9768((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9769BDBM9769((2S)-2-[(4-methylbenzene)(2-methylpropyl)sulfonami...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9771BDBM9771((2S)-6-(2-benzyl-3,3-dimethylbutanamido)-2-[(4-met...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Pharmacor

LigandChemical structure of BindingDB Monomer ID 9772BDBM9772((2S)-6-{[(benzyloxy)carbonyl]amino}-2-[(4-methylbe...)
Affinity DataKi: >300nM ΔG°: >-37.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2006
Entry Details Article
PubMed