Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50014164
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138941(Methyl-[3-phenyl-2-m-tolyl-2H-[1,2,4]thiadiazol-(5...)
Affinity DataEC50:  640nMAssay Description:Effective concentration for displacement of [3H]CCPA from human A1 adenosine receptor after 60 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138944([2,3-Di-p-tolyl-2H-[1,2,4]thiadiazol-(5E)-ylidene]...)
Affinity DataEC50:  1.60E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138943([2-(4-Methoxy-phenyl)-3-phenyl-2H-[1,2,4]thiadiazo...)
Affinity DataEC50:  2.40E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM60981(SCH-202676 hydrobromide | SMR001230740 | MLS002153...)
Affinity DataEC50:  2.80E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed