Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50014164
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM60981((2,3-diphenyl-1,2,4-thiadiazol-5-ylidene)-methyl-a...)
Affinity DataEC50:  2.80E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138944(CHEMBL351194 | [2,3-Di-p-tolyl-2H-[1,2,4]thiadiazo...)
Affinity DataEC50:  1.60E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138941(CHEMBL351012 | Methyl-[3-phenyl-2-m-tolyl-2H-[1,2,...)
Affinity DataEC50:  640nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human A1 adenosine receptor after 60 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50138943(CHEMBL161767 | [2-(4-Methoxy-phenyl)-3-phenyl-2H-[...)
Affinity DataEC50:  2.40E+3nMAssay Description:Effective concentration for displacement of [3H]-CCPA from human adenosine A1 receptor after 60 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed