Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50014238
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139872(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139876(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139869(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139871(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018152(CHEMBL274855 | 8-Phenyl-1-propyl-3,7-dihydro-purin...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]ZM-241385 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139869(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139874(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139878(4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139875(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139877(4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  10nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50110985(1-Butyl-8-phenyl-3,7-dihydro-purine-2,6-dione | CH...)
Affinity DataKi:  11.8nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]ZM-241385 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139875(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  13nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139876(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139873(4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  18.9nMAssay Description:Binding affinity for human HEK293 adenosine A2B receptor using [125I]ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139879(4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139874(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139874(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  23nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139872(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  26nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139871(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139878(4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50110985(1-Butyl-8-phenyl-3,7-dihydro-purine-2,6-dione | CH...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139871(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  43nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  53.4nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]ZM-241385 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139875(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139873(4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018152(CHEMBL274855 | 8-Phenyl-1-propyl-3,7-dihydro-purin...)
Affinity DataKi:  67nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139870(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  70nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]ZM-241385 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139869(4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139872(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  89nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139877(4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139879(4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(CHEMBL418333 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataKi:  183nMAssay Description:Binding affinity for human adenosine A3 receptor using [3H]-PBS-11 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  190nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(CHEMBL418333 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataKi:  210nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(CHEMBL418333 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataKi:  250nMAssay Description:Binding affinity for human adenosine A2B receptor using [3H]-PSB-298 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018157(CHEMBL9069 | 1-Methyl-8-phenyl-3,7-dihydro-purine-...)
Affinity DataKi:  260nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  415nMAssay Description:Binding affinity for human HEK293 adenosine A2B receptor using [125I]ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139870(4-(1-Butyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8...)
Affinity DataKi:  475nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50110985(1-Butyl-8-phenyl-3,7-dihydro-purine-2,6-dione | CH...)
Affinity DataKi:  642nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor of rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  850nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139868(4-(1-Methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]-CCPA from adenosine A1 receptor of rat brain cortical membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM82023(4-(1,3-Dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  1.33E+3nMAssay Description:Binding affinity for human HEK293 adenosine A2B receptor using [125I]ABOPX in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018162(CHEMBL418333 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018152(CHEMBL274855 | 8-Phenyl-1-propyl-3,7-dihydro-purin...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50042209(4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-...)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]PIA in rat brain cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50018157(CHEMBL9069 | 1-Methyl-8-phenyl-3,7-dihydro-purine-...)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50139871(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity for human adenosine A3 receptor using [3H]PBS-11 in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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