Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50036084
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004276BDBM50004276(CHEMBL111448 | 1-Isopropyl-2-oxo-1,2-dihydro-quino...)
Affinity DataKi:  0.0320nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004292BDBM50004292(CHEMBL148076 | 2-Isopropoxy-quinoline-4-carboxylic...)
Affinity DataKi:  0.310nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004279BDBM50004279(CHEMBL148430 | 2-Propoxy-quinoline-4-carboxylic ac...)
Affinity DataKi:  0.320nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004288BDBM50004288(CHEMBL111059 | 2-Butoxy-quinoline-4-carboxylic aci...)
Affinity DataKi:  0.390nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004284BDBM50004284(CHEMBL113742 | 2-Isobutoxy-quinoline-4-carboxylic ...)
Affinity DataKi:  0.440nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004268BDBM50004268(CHEMBL325349 | 2-Oxo-1-propyl-1,2-dihydro-quinolin...)
Affinity DataKi:  0.450nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004297BDBM50004297(CHEMBL113519 | 1-Isobutyl-2-oxo-1,2-dihydro-quinol...)
Affinity DataKi:  0.470nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004278BDBM50004278(CHEMBL333371 | 2-Oxo-1-phenyl-1,2-dihydro-quinolin...)
Affinity DataKi:  0.510nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004286BDBM50004286(CHEMBL112941 | 2-Methoxy-quinoline-4-carboxylic ac...)
Affinity DataKi:  0.580nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004287BDBM50004287(CHEMBL112237 | 1-Butyl-2-oxo-1,2-dihydro-quinoline...)
Affinity DataKi:  0.680nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004295BDBM50004295(CHEMBL321477 | 2-Pentyloxy-quinoline-4-carboxylic ...)
Affinity DataKi:  0.860nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004282BDBM50004282(CHEMBL325235 | 2-Ethoxy-quinoline-4-carboxylic aci...)
Affinity DataKi:  0.880nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004296BDBM50004296(CHEMBL113204 | 2-Oxo-1-pentyl-1,2-dihydro-quinolin...)
Affinity DataKi:  0.960nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004273BDBM50004273(CHEMBL322751 | 1-Ethyl-2-oxo-1,2-dihydro-quinoline...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004300BDBM50004300(CHEMBL112224 | 1-Hexyl-2-oxo-1,2-dihydro-quinoline...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004266BDBM50004266(CHEMBL114444 | 1-Benzyl-2-oxo-1,2-dihydro-quinolin...)
Affinity DataKi:  1.30nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004291BDBM50004291(CHEMBL326545 | 1-(3-Methyl-butyl)-2-oxo-1,2-dihydr...)
Affinity DataKi:  1.5nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000483BDBM50000483(CHEMBL519643 | 1-Methyl-1H-indazole-3-carboxylic a...)
Affinity DataKi:  2.10nMAssay Description:Compound was evaluated for its ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15. More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004299BDBM50004299(CHEMBL419012 | 1-Methyl-2-oxo-1,2-dihydro-quinolin...)
Affinity DataKi:  2.60nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004271BDBM50004271(CHEMBL423687 | 2-Hexyloxy-quinoline-4-carboxylic a...)
Affinity DataKi:  3.20nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004275BDBM50004275(CHEMBL148398 | 2-Oxo-1,2-dihydro-quinoline-4-carbo...)
Affinity DataKi:  4.40nMAssay Description:Compound was evaluated for its ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15. More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004290BDBM50004290(CHEMBL147262 | Quinoline-4-carboxylic acid 8-methy...)
Affinity DataKi:  7.10nMAssay Description:Compound was evaluated for its ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15. More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 85330BDBM85330(NSC_68647 | CAS_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  7.60nMAssay Description:Compound was evaluated for its ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15. More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004294BDBM50004294(CHEMBL424117 | 1-Butyl-2-oxo-1,2,3,4-tetrahydro-qu...)
Affinity DataKi:  8.70nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004285BDBM50004285(CHEMBL114080 | 2-Butoxy-quinoline-4-carboxylic aci...)
Affinity DataKi:  19nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004289BDBM50004289(CHEMBL109813 | 2-Propoxy-quinoline-4-carboxylic ac...)
Affinity DataKi:  42nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004293BDBM50004293(CHEMBL144560 | 1-Butyl-6-methyl-2-oxo-1,2-dihydro-...)
Affinity DataKi:  44nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004298BDBM50004298(CHEMBL332037 | 2-Isopropoxy-quinoline-4-carboxylic...)
Affinity DataKi:  53nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004281BDBM50004281(CHEMBL324243 | 1-Butyl-2-oxo-1,2-dihydro-quinoline...)
Affinity DataKi:  60nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004272BDBM50004272(CHEMBL112942 | 2-Oxo-1-phenyl-1,2-dihydro-quinolin...)
Affinity DataKi:  63nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004267BDBM50004267(CHEMBL113118 | 2-Oxo-1-propyl-1,2-dihydro-quinolin...)
Affinity DataKi:  67nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004280BDBM50004280(CHEMBL434652 | Quinoline-4-carboxylic acid (8-meth...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004270BDBM50004270(CHEMBL148209 | 1-Methyl-2-oxo-1,2-dihydro-quinolin...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004283BDBM50004283(CHEMBL342574 | 1-Butyl-3-ethyl-2-oxo-1,2-dihydro-q...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004277BDBM50004277(CHEMBL343836 | 2-Oxo-1,2-dihydro-quinoline-4-carbo...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004274BDBM50004274(CHEMBL359246 | 1-Butyl-3-ethyl-2-oxo-1,2-dihydro-q...)
Affinity DataKi:  160nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed