Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50037293
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141067BDBM50141067(3-[4-(2,4-Difluoro-phenoxy)-phenyl]-pyrazole-1-car...)
Affinity DataKi:  25nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141062BDBM50141062(3-[4-(4-Fluoro-phenoxy)-phenyl]-pyrazole-1-carboxy...)
Affinity DataKi:  31nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141070BDBM50141070(3-[4-(4-Nitro-phenoxy)-phenyl]-pyrazole-1-carboxyl...)
Affinity DataKi:  31nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141072BDBM50141072(3-(4-Phenoxy-phenyl)-pyrazole-1-carboxylic acid am...)
Affinity DataKi:  35nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141065BDBM50141065(3-[4-(4-Fluoro-phenoxy)-phenyl]-pyrazole-1-carboxy...)
Affinity DataKi:  150nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141073BDBM50141073((E)-2-(4-(4-fluorophenoxy)benzylidene)hydrazinecar...)
Affinity DataKi:  180nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141066BDBM50141066(3-[4-(4-Fluoro-phenoxy)-phenyl]-1H-pyrazole | CHEM...)
Affinity DataKi:  200nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141064BDBM50141064(3-(4-Phenoxy-phenyl)-1H-pyrazole | CHEMBL41864)
Affinity DataKi:  240nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141071BDBM50141071(3-[4-(4-Fluoro-phenoxy)-phenyl]-pyrazole-1-carboxy...)
Affinity DataKi:  340nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141069BDBM50141069(3-[4-(4-Fluoro-phenoxy)-phenyl]-1-methyl-1H-pyrazo...)
Affinity DataKi:  690nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031299BDBM50031299(CHEMBL741 | BW-430C | 6-(2,3-Dichloro-phenyl)-[1,2...)
Affinity DataKi:  1.70E+4nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003655BDBM50003655(Phenytoin)
Affinity DataKi:  2.40E+4nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50003659BDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...)
Affinity DataKi:  5.20E+4nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078831BDBM50078831(3-Phenyl-1H-pyrazole | CHEMBL38876)
Affinity DataKi:  6.10E+4nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSodium channel protein type 4 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141063BDBM50141063(3-(4-Methoxy-phenyl)-1H-pyrazole | CHEMBL39210)
Affinity DataKi:  8.10E+4nMAssay Description:Affinity for inactive human SkM1 sodium channel expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed