Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50041077
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142344((S)-3-(6-Methoxy-pyridin-3-yl)-3-{methyl-[5-(3-met...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142341((S)-3-(6-Methoxy-pyridin-3-yl)-3-{methyl-[5-(3-vin...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142342((S)-3-{[5-(3-Amino-5,6,7,8-tetrahydro-[1,8]naphthy...)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142338((S)-3-{[5-(3-Acetylamino-5,6,7,8-tetrahydro-[1,8]n...)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142343((S)-3-(6-Methoxy-pyridin-3-yl)-3-[methyl-(5-5,6,7,...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142336((S)-3-{[5-(3-Methanesulfonylamino-5,6,7,8-tetrahyd...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142340((S)-3-(6-Methoxy-pyridin-3-yl)-3-{methyl-[5-(3-phe...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142337((S)-3-{[5-(3-Bromo-5,6,7,8-tetrahydro-[1,8]naphthy...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142339((S)-3-{[5-(3-Cyano-5,6,7,8-tetrahydro-[1,8]naphthy...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50142345((S)-3-(6-Methoxy-pyridin-3-yl)-3-{methyl-[5-(3-nit...)
Affinity DataIC50:  37nMAssay Description:Displacement of [125I]L-775,219 from human recombinant alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed