Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50000341
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004610(2-(2-{2-[2-(2-{[1-(2-Acetylamino-3-hydroxy-propion...)
Affinity DataKi:  1.01E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004613(1-(2-Acetylamino-3-hydroxy-propionyl)-pyrrolidine-...)
Affinity DataKi:  1.35E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004609(2-{2-[2-(2-{2-[(1-Acetyl-pyrrolidine-2-carbonyl)-a...)
Affinity DataKi:  1.67E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004605(1-(2-Acetylamino-3-hydroxy-propionyl)-pyrrolidine-...)
Affinity DataKi:  2.23E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004611(2-(2-{2-[2-(2-Acetylamino-3-phenyl-propionylamino)...)
Affinity DataKi:  2.30E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004607(1-Acetyl-pyrrolidine-2-carboxylic acid (1-{1-[1-(1...)
Affinity DataKi:  2.66E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004606(2-(2-Acetylamino-3-phenyl-propionylamino)-5-guanid...)
Affinity DataKi:  4.79E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004614(1-Acetyl-pyrrolidine-2-carboxylic acid {1-[1-(1-ca...)
Affinity DataKi:  5.78E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004604(2-(2-Acetylamino-3-phenyl-propionylamino)-5-guanid...)
Affinity DataKi:  7.18E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004608(2-{2-[2-(2-Acetylamino-5-guanidino-pentanoylamino)...)
Affinity DataKi:  9.50E+5nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein(Sus scrofa)
University Hospital

Curated by ChEMBL
LigandPNGBDBM50004612(1-(2-Acetylamino-3-hydroxy-propionyl)-pyrrolidine-...)
Affinity DataKi:  2.29E+6nMAssay Description:Inhibitory activity against beta-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed